6833 |
ATP BINDING CASSETTE SUBFAMILY C MEMBER 8 |
ABCC8 |
ABC36 |
HHF1 |
HI |
HRINS |
MRP8 |
PHHI |
SUR |
SUR1 |
SUR1delta2 |
TNDM2 |
600509 |
59 |
ENSG00000006071 |
OTTHUMG00000166316 |
SULFONYLUREA RECEPTOR 1. [SOURCE:UNIPROT/SWISSPROT;ACC:Q09428] |
Q09428 |
ATP-BINDING CASSETTE SUB-FAMILY C MEMBER 8 |
ABCC8_HUMAN |
Sulfonylurea receptor 1 |
PA24395 |
ATP-binding cassette transporter C8 |
T91480 |
PNDM3 |
Human Readable Name | DRUGGABLE GENOME |
Interpro Short Name | ABC_transptr_TM_dom |
Interpro Acc | IPR001140 |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | ABC TRANSPORTER |
Interpro Name | ABC transporter, transmembrane domain |
Uniprot Status | Swiss-Prot |
Interpro Type | Domain |
Target Class | Transporters |
Target Subclass | TC:3.A.1.208.4 |
Gene Biotype | PROTEIN_CODING |
TRANSPORTER |
ABC TRANSPORTER |
DRUGGABLE GENOME |
inhibitor (inhibitory) |
Novel drug target | Established target |
Trial Name | mitiglinide, KAD-1229,Glufast, Glinsuna, Metgluna |
blocker (inhibitory) |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
Trial Name | Starlix |
blocker (inhibitory) |
inducer (activating) |
Trial Name | glimepiride,Amaryl |
Novel drug target | Established target |
Trial Name | rosiglitazone + glimepiride,Avandaryl |
blocker (inhibitory) |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Novel drug target | Established target |
Trial Name | glyburide + metformin,Glucovance |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
blocker (inhibitory) |
inhibitor (inhibitory) |
Novel drug target | Established target |
Trial Name | repaglinide,Prandin, NovoNorm, PrandiMet |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
blocker (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
blocker (inhibitory) |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
Direct Interaction | yes |
blocker (inhibitory) |
inhibitor (inhibitory) |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
Direct Interaction | yes |
n/a |
Mechanism of Interaction | Sulfonylurea receptors; K-ATP channels opener |
Direct Interaction | yes |
n/a |
Mechanism of Interaction | Sulfonylurea receptors; K-ATP channels opener |
Direct Interaction | yes |
blocker (inhibitory) |
inhibitor (inhibitory) |
Mechanism of Interaction | Sulfonylurea receptor 1, Kir6.2 blocker |
Direct Interaction | yes |
ABCC8 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ABCC8 | Display Id |
ENSG00000006071 | Ensembl Gene Id |
SULFONYLUREA RECEPTOR 1. [SOURCE:UNIPROT/SWISSPROT;ACC:Q09428] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
ABCC8 | Gene Symbol |
Target Class | Transporters |
Target Subclass | TC:3.A.1.208.4 |
ABCC8_HUMAN | Uniprot Id |
Q09428 | Uniprot Accession |
ENSG00000006071 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
Interpro Short Name | ABC_transptr_TM_dom |
Interpro Acc | IPR001140 |
ABC TRANSPORTER, DRUGGABLE GENOME |
PA24395 | PharmGKB ID |
ENSG00000006071 | Gene Symbol |
ABCC8 | Ensembl Id |
DRUGGABLE GENOME |
SUR | GENE_SYMBOL |
SUR1 | GENE_SYMBOL |
ABCC8 | GENE_SYMBOL |
HRINS | GO Gene Synonym |
SUR | GO Gene Synonym |
SUR1 | GO Gene Synonym |
ABC TRANSPORTER |
ABCC8 | TTD Gene Abbreviation |
T91480 | TTD Target ID |
ATP-binding cassette sub-family C member 8 | Gene Name |
Q09428 | UniProt ID |
TRANSPORTER |