94 |
ACTIVIN A RECEPTOR LIKE TYPE 1 |
ACVRL1 |
ACVRLK1 |
ALK-1 |
ALK1 |
HHT |
HHT2 |
ORW2 |
SKR3 |
TSR-I |
601284 |
175 |
ENSG00000139567 |
OTTHUMG00000169507 |
ACTIVIN RECEPTOR-LIKE KINASE 1 |
ACTIVIN RECEPTOR-LIKE KINASE-1 |
TGF-B SUPERFAMILY RECEPTOR TYPE I |
SERINE/THREONINE-PROTEIN KINASE RECEPTOR R3 |
P37023 |
SERINE/THREONINE-PROTEIN KINASE RECEPTOR R3 PRECURSOR (EC 2.7.1.37) (SKR3) (ACTIVIN RECEPTOR-LIKE KINASE 1) (ALK-1) (TGF-B SUPERFAMILY RECEPTOR TYPE I) (TSR-I). [SOURCE:UNIPROT/SWISSPROT;ACC:P37023] |
T36959 |
Target Subclass | EC:2.7.11.30 |
Target Class | Receptors |
Human Readable Name | DRUGGABLE GENOME |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
KINASE |
SERINE THREONINE KINASE |
DRUGGABLE GENOME |
ENZYME |
inhibitor (inhibitory) |
Mechanism of Interaction | Serine/threonine-protein kinase receptor R3 inhibitor |
Direct Interaction | yes |
n/a |
Trial Name | ACE-041 |
Novel drug target | Novel Target |
inhibitor (inhibitory) |
Mechanism of Interaction | Serine/threonine-protein kinase receptor R3 inhibitor |
Direct Interaction | yes |
ACVRL1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
SERINE/THREONINE-PROTEIN KINASE RECEPTOR R3 PRECURSOR (EC 2.7.1.37) (SKR3) (ACTIVIN RECEPTOR-LIKE KINASE 1) (ALK-1) (TGF-B SUPERFAMILY RECEPTOR TYPE I) (TSR-I). [SOURCE:UNIPROT/SWISSPROT;ACC:P37023] | Description |
ENSG00000139567 | Ensembl Gene Id |
ACVRL1 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
ACVRL1 | Gene Symbol |
Target Class | Receptors |
Target Subclass | EC:2.7.11.30 |
ACVRL1 | TTD Gene Abbreviation |
T36959 | TTD Target ID |
ALK1 | GENE_SYMBOL |
ACVRL1 | GENE_SYMBOL |
Serine/threonine-protein kinase receptor R3 | UNIPROT |
ENSG00000139567 | Gene Symbol |
ACVRL1 | Ensembl Id |
DRUGGABLE GENOME |
ENSG00000139567 | Ensembl Gene ID |
ACVRLK1 | Human Protein Atlas Gene Synonym |
ALK1 | Human Protein Atlas Gene Synonym |
ENZYME |
ACVRLK1 | GO Gene Synonym |
ALK1 | GO Gene Synonym |
CELL SURFACE, SERINE THREONINE KINASE |
94 | Gene ID |
ACVRLK1 | dGene Synonym |
ALK-1 | dGene Synonym |
KINASE, SERINE THREONINE KINASE |
Serine/threonine-protein kinase receptor R3 | Gene Name |
P37023 | UniProt ID |
KINASE |