23621 |
BETA-SECRETASE 1 |
BACE1 |
ASP2 |
BACE |
HSPC104 |
604252 |
933 |
ENSG00000186318 |
OTTHUMG00000160636 |
KIAA1149 |
BACE1_HUMAN |
P56817 |
Aspartyl protease 2 |
Beta-site amyloid precursor protein cleaving enzyme 1 |
Memapsin-2 |
Membrane-associated aspartic protease 2 |
Asp 2 |
Beta-site APP cleaving enzyme 1 |
BETA-SECRETASE 1 PRECURSOR (EC 3.4.23.46) (BETA-SITE APP CLEAVING ENZYME 1) (BETA-SITE AMYLOID PRECURSOR PROTEIN CLEAVING ENZYME 1) (ASPARTYL PROTEASE 2) (ASP 2) (ASP2) (MEMBRANE-ASSOCIATED ASPARTIC PROTEASE 2) (MEMAPSIN-2). [SOURCE:UNIPROT/SWISSPROT;ACC: |
BETA-SECRETASE |
T79031 |
T73992 |
Human Readable Name | PROTEASE |
Target Class | Enzymes |
Target Subclass | EC:3.4.23.46 |
Human Readable Name | DRUGGABLE GENOME |
Interpro Name | Peptidase aspartic, active site |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Peptidase_aspartic_AS |
Interpro Type | Active_site |
Interpro Acc | IPR001969 |
Uniprot Status | Swiss-Prot |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
PROTEASE |
DRUGGABLE GENOME |
inhibitor (inhibitory) |
Mechanism of Interaction | Beta-secretase 1 inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
n/a |
Trial Name | [(+)-phenserine tartrate,Posiphen |
Novel drug target | Novel Target |
Trial Name | Posiphen |
BACE1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
BACE1 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:3.4.23.46 |
ENSG00000186318 | Ensembl Gene Id |
BETA-SECRETASE 1 PRECURSOR (EC 3.4.23.46) (BETA-SITE APP CLEAVING ENZYME 1) (BETA-SITE AMYLOID PRECURSOR PROTEIN CLEAVING ENZYME 1) (ASPARTYL PROTEASE 2) (ASP 2) (ASP2) (MEMBRANE-ASSOCIATED ASPARTIC PROTEASE 2) (MEMAPSIN-2). [SOURCE:UNIPROT/SWISSPROT;ACC: | Description |
BACE1 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
BACE1 | Uniprot Gene Name |
P56817 | Uniprot Accession |
BACE1_HUMAN | Uniprot Id |
Interpro Name | Peptidase aspartic, active site |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Peptidase_aspartic_AS |
PROTEASE, DRUGGABLE GENOME |
BACE | TTD Gene Abbreviation |
T73992 | TTD Target ID |
ENSG00000186318 | Gene Symbol |
BACE1 | Ensembl Id |
DRUGGABLE GENOME |
KIAA1149 | GENE_SYMBOL |
BACE1 | GENE_SYMBOL |
Beta-secretase 1 | UNIPROT |
BACE | GO Gene Synonym |
KIAA1149 | GO Gene Synonym |
CELL SURFACE, PROTEASE |
23621 | Gene ID |
ASP2 | dGene Synonym |
BACE | dGene Synonym |
PROTEASE |
BACE1 | TTD Gene Abbreviation |
T79031 | TTD Target ID |