624 |
BRADYKININ RECEPTOR B2 |
BDKRB2 |
B2R |
BK-2 |
BK2 |
BKR2 |
BRB2 |
113503 |
1030 |
ENSG00000168398 |
OTTHUMG00000171408 |
P30411 |
BKRB2_HUMAN |
B2 bradykinin receptor |
BK-2 receptor |
PA80 |
B2 BRADYKININ RECEPTOR (BK-2 RECEPTOR) (B2R). [SOURCE:UNIPROT/SWISSPROT;ACC:P30411] |
T23714 |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Interpro Type | Family |
Interpro Acc | IPR000276 |
Uniprot Status | Swiss-Prot |
Gene Biotype | PROTEIN_CODING |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Trial Name | Firazyr, icatibant, JE049 |
Novel drug target | Established target |
agonist (activating) |
Mechanism of Interaction | Bradykinin B2 receptor agonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Bradykinin B2 receptor antagonist |
Direct Interaction | yes |
Trial Name | anatibant |
antagonist (inhibitory) |
Mechanism of Interaction | Bradykinin B2 receptor antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Bradykinin B2 receptor antagonist |
Direct Interaction | yes |
agonist (activating) |
BDKRB2 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
BDKRB2 | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
B2 BRADYKININ RECEPTOR | Uniprot Protein Name |
ENSG00000168398 | Ensembl Gene Id |
BDKRB2 | Uniprot Gene Name |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
BDKRB2 | Gene Symbol |
ENSG00000168398 | Ensembl Gene Id |
P30411 | Uniprot Accession |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
B2 BRADYKININ RECEPTOR (BK-2 RECEPTOR) (B2R). [SOURCE:UNIPROT/SWISSPROT;ACC:P30411] | Description |
BDKRB2 | Display Id |
ENSG00000168398 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PA80 | PharmGKB ID |
BKR2 | GENE_SYMBOL |
BDKRB2 | GENE_SYMBOL |
B2 bradykinin receptor | UNIPROT |
ENSG00000168398 | Gene Symbol |
BDKRB2 | Ensembl Id |
DRUGGABLE GENOME |
BKR2 | GO Gene Synonym |
G PROTEIN COUPLED RECEPTOR |
624 | Gene ID |
B2R | dGene Synonym |
BK-2 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
BDKRB2 | TTD Gene Abbreviation |
T23714 | TTD Target ID |