773 |
CALCIUM VOLTAGE-GATED CHANNEL SUBUNIT ALPHA1 A |
CACNA1A |
APCA |
BI |
CACNL1A4 |
CAV2.1 |
EA2 |
EIEE42 |
FHM |
HPCA |
MHP |
MHP1 |
SCA6 |
601011 |
1388 |
ENSG00000141837 |
OTTHUMG00000044590 |
Voltage-gated calcium channel subunit alpha Cav2.1 |
Calcium channel, L type, alpha-1 polypeptide isoform 4 |
Brain calcium channel I |
Voltage-dependent P/Q-type calcium channel subunit alpha-1A |
CACN3 |
O00555 |
CAC1A_HUMAN |
CACH4 |
PA26007 |
VOLTAGE-DEPENDENT P/Q-TYPE CALCIUM CHANNEL ALPHA-1A SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV2.1) (CALCIUM CHANNEL, L TYPE, ALPHA-1 POLYPEPTIDE ISOFORM 4) (BRAIN CALCIUM CHANNEL I) (BI). [SOURCE:UNIPROT/SWISSPROT;ACC:O00555] |
Voltage-gated calcium channel alpha Cav2.1 |
T34949 |
DEE42 |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11 |
Target Subclass | Channels |
Target Main Class | Transporters |
Target Subclass | CalciumChannels |
Transmembrane Helix Count | 23 |
Target Subclass | Voltage_gated_ion_channels |
Initial Gene Query | Cav2.1 |
Counted Citations from 1950-2000 | 714 |
Human Readable Name | DRUGGABLE GENOME |
Interpro Short Name | Ion_trans_dom |
Interpro Type | Domain |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR005821 |
Uniprot Status | Swiss-Prot |
Interpro Name | Ion transport domain |
Human Readable Name | ION CHANNEL |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
inhibitor (inhibitory) |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
Trial Name | pregabalin,Lyrica |
n/a |
Trial Name | - |
Novel drug target | Established target |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated P/Q-type calcium channel alpha-1A subunit blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated calcium channel blocker |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
CACNA1A | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
CAC1A_HUMAN | Uniprot Id |
ENSG00000141837 | Ensembl Gene Id |
O00555 | Uniprot Accession |
Target Subclass | Channels |
Target Main Class | Transporters |
Target Subclass | CalciumChannels |
773 | Entrez Gene ID |
Initial Gene Query | Cav2.1 |
Counted Citations from 1950-2000 | 714 |
ION CHANNEL |
O00555 | Uniprot Accession |
VOLTAGE-DEPENDENT P/Q-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1A | Uniprot Protein Name |
CAC1A_HUMAN | Uniprot Id |
Interpro Type | Domain |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR005821 |
ION CHANNEL, DRUGGABLE GENOME |
CACNA1A | Display Id |
ENSG00000141837 | Ensembl Gene Id |
VOLTAGE-DEPENDENT P/Q-TYPE CALCIUM CHANNEL ALPHA-1A SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV2.1) (CALCIUM CHANNEL, L TYPE, ALPHA-1 POLYPEPTIDE ISOFORM 4) (BRAIN CALCIUM CHANNEL I) (BI). [SOURCE:UNIPROT/SWISSPROT;ACC:O00555] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
CACNA1A | Gene Symbol |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11 |
PA26007 | PharmGKB ID |
ENSG00000141837 | Gene Symbol |
CACNA1A | Ensembl Id |
DRUGGABLE GENOME |
CACN3 | GENE_SYMBOL |
CACNL1A4 | GENE_SYMBOL |
CACNA1A | GENE_SYMBOL |
CACNA1A | TTD Gene Abbreviation |
T34949 | TTD Target ID |
Voltage-dependent P/Q-type calcium channel subunit alpha-1A | Gene Name |
O00555 | UniProt ID |
ION CHANNEL |