774 |
CALCIUM VOLTAGE-GATED CHANNEL SUBUNIT ALPHA1 B |
CACNA1B |
BIII |
CACNL1A5 |
CACNN |
Cav2.2 |
DYT23 |
601012 |
1389 |
ENSG00000148408 |
OTTHUMG00000021002 |
VOLTAGE-DEPENDENT N-TYPE CALCIUM CHANNEL ALPHA-1B SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV2.2) (CALCIUM CHANNEL, L TYPE, ALPHA-1 POLYPEPTIDE ISOFORM 5) (BRAIN CALCIUM CHANNEL III) (BIII). [SOURCE:UNIPROT/SWISSPROT;ACC:Q00975] |
Q00975 |
CAC1B_HUMAN |
Voltage-gated calcium channel subunit alpha Cav2.2 |
Calcium channel, L type, alpha-1 polypeptide isoform 5 |
Brain calcium channel III |
Voltage-dependent N-type calcium channel subunit alpha-1B |
CACH5 |
PA26008 |
Voltage-gated calcium channel alpha Cav2.2 |
T38338 |
NEDNEH |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11 |
Target Subclass | Channels |
Target Subclass | CalciumChannels |
Transmembrane Helix Count | 22 |
Target Subclass | Voltage_gated_ion_channels |
Target Main Class | Transporters |
Human Readable Name | ION CHANNEL |
Uniprot Status | Swiss-Prot |
Interpro Name | Ion transport domain |
Interpro Acc | IPR005821 |
Interpro Type | Domain |
Interpro Short Name | Ion_trans_dom |
Uniprot Evidence | 1: Evidence at protein level |
Initial Gene Query | Cav2.2 |
Counted Citations from 1950-2000 | 290 |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
blocker (inhibitory) |
Trial Name | CNV2197944 |
Novel drug target | Established target |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
Direct Interaction | yes |
blocker (inhibitory) |
inhibitor (inhibitory) |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
Direct Interaction | yes |
Trial Name | levetiracetam ,Keppra, Keppra XR |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
Direct Interaction | yes |
inhibitor (inhibitory) |
modulator |
Direct Interaction | yes |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Trial Name | Depomed |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated N-type calcium channel alpha-1B subunit blocker |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
Trial Name | XP13512 |
n/a |
Novel drug target | Established target |
Trial Name | Safinamide |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated calcium channel blocker |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Direct Interaction | yes |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
CACNA1B | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
CACNA1B | Display Id |
ENSG00000148408 | Ensembl Gene Id |
VOLTAGE-DEPENDENT N-TYPE CALCIUM CHANNEL ALPHA-1B SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV2.2) (CALCIUM CHANNEL, L TYPE, ALPHA-1 POLYPEPTIDE ISOFORM 5) (BRAIN CALCIUM CHANNEL III) (BIII). [SOURCE:UNIPROT/SWISSPROT;ACC:Q00975] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
CACNA1B | Gene Symbol |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11 |
CACNA1B | Gene Symbol |
CAC1B_HUMAN | Uniprot Id |
774 | Entrez Gene Id |
Target Subclass | Channels |
Target Subclass | CalciumChannels |
Transmembrane Helix Count | 22 |
VOLTAGE-DEPENDENT N-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1B | Uniprot Protein Name |
CAC1B_HUMAN | Uniprot Id |
Q00975 | Uniprot Accession |
Human Readable Name | ION CHANNEL |
Uniprot Status | Swiss-Prot |
Human Readable Name | DRUGGABLE GENOME |
ION CHANNEL, DRUGGABLE GENOME |
774 | Entrez Gene ID |
Initial Gene Query | Cav2.2 |
Counted Citations from 1950-2000 | 290 |
ION CHANNEL |
PA26008 | PharmGKB ID |
ENSG00000148408 | Gene Symbol |
CACNA1B | Ensembl Id |
DRUGGABLE GENOME |
CACNL1A5 | GENE_SYMBOL |
CACNA1B | GENE_SYMBOL |
Voltage-dependent N-type calcium channel subunit alpha-1B | UNIPROT |
CACNA1B | TTD Gene Abbreviation |
T38338 | TTD Target ID |
Voltage-dependent N-type calcium channel subunit alpha-1B | Gene Name |
Q00975 | UniProt ID |
ION CHANNEL |