834 |
CASPASE 1 |
CASP1 |
ICE |
IL1BC |
P45 |
147678 |
1499 |
ENSG00000137752 |
OTTHUMG00000048072 |
P29466 |
CASPASE-1 SUBUNIT P20 |
CASP1_HUMAN |
IL1BCE |
CASPASE-1 PRECURSOR (EC 3.4.22.36) (CASP-1) (INTERLEUKIN-1 BETA CONVERTASE) (IL-1BC) (IL-1 BETA CONVERTING ENZYME) (ICE) (INTERLEUKIN- 1 BETA CONVERTING ENZYME) (P45). [SOURCE:UNIPROT/SWISSPROT;ACC:P29466] |
IL-1 beta-converting enzyme |
IL-1BC |
CASP-1 |
Interleukin-1 beta-converting enzyme |
Interleukin-1 beta convertase |
Caspase-1 subunit p10 |
Caspase-1 |
T98269 |
Human Readable Name | PROTEASE |
Interpro Acc | IPR002398 |
Interpro Name | Peptidase C14, caspase precursor p45 |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Pept_C14_p45 |
Uniprot Status | Swiss-Prot |
Interpro Type | Family |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Enzymes |
Target Subclass | EC:3.4.22.36 |
Gene Biotype | PROTEIN_CODING |
PROTEASE |
DRUGGABLE GENOME |
ENZYME |
n/a |
Trial Name | VX-765 |
Novel drug target | Novel Target |
inhibitor (inhibitory) |
Mechanism of Interaction | Caspase-1 inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Caspase inhibitor |
Direct Interaction | yes |
CASP1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000137752 | Ensembl Gene Id |
CASPASE-1 PRECURSOR (EC 3.4.22.36) (CASP-1) (INTERLEUKIN-1 BETA CONVERTASE) (IL-1BC) (IL-1 BETA CONVERTING ENZYME) (ICE) (INTERLEUKIN- 1 BETA CONVERTING ENZYME) (P45). [SOURCE:UNIPROT/SWISSPROT;ACC:P29466] | Description |
CASP1 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
CASP1 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:3.4.22.36 |
834 | Entrez Gene Id |
CASP1 | Uniprot Gene Name |
CASP1_HUMAN | Uniprot Id |
Interpro Acc | IPR002398 |
Interpro Name | Peptidase C14, caspase precursor p45 |
Uniprot Evidence | 1: Evidence at protein level |
PROTEASE, DRUGGABLE GENOME |
ENSG00000137752 | Gene Symbol |
CASP1 | Ensembl Id |
DRUGGABLE GENOME |
IL1BCE | GENE_SYMBOL |
CASP1 | GENE_SYMBOL |
Caspase-1 | UNIPROT |
834 | Gene ID |
ICE | dGene Synonym |
IL1BC | dGene Synonym |
PROTEASE |
CASP1 | TTD Gene Abbreviation |
T98269 | TTD Target ID |
Caspase-1 | Gene Name |
P29466 | UniProt ID |
ENZYME |