846 |
CALCIUM SENSING RECEPTOR |
CASR |
CAR |
EIG8 |
FHH |
FIH |
GPRC2A |
HHC |
HHC1 |
HYPOC1 |
NSHPT |
PCAR1 |
hCasR |
601199 |
1514 |
ENSG00000036828 |
P41180 |
EXTRACELLULAR CALCIUM-SENSING RECEPTOR |
EXTRACELLULAR CALCIUM-SENSING RECEPTOR PRECURSOR (CASR) (PARATHYROID CELL CALCIUM-SENSING RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P41180] |
CASR_HUMAN |
Parathyroid cell calcium-sensing receptor 1 |
PA26097 |
T92076 |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Glutamate |
Human Readable Name | DRUGGABLE GENOME |
Interpro Acc | IPR000337 |
Interpro Type | Family |
Interpro Name | GPCR, family 3 |
Uniprot Status | Swiss-Prot |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Short Name | GPCR_3 |
Uniprot Evidence | 1: Evidence at protein level |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
allosteric modulator |
antagonist (inhibitory) |
Mechanism of Interaction | Calcium sensing receptor antagonist |
Direct Interaction | yes |
Trial Name | ronacaleret, 751689 |
agonist (activating) |
Mechanism of Interaction | Calcium sensing receptor agonist |
Direct Interaction | yes |
positive modulator (activating) |
Mechanism of Interaction | Calcium sensing receptor positive allosteric modulator |
Direct Interaction | yes |
n/a |
Trial Name | NPS-2143 |
Novel drug target | Established target |
modulator |
Mechanism of Interaction | Calcium sensing receptor modulator |
Direct Interaction | yes |
positive modulator (activating) |
Mechanism of Interaction | Calcium sensing receptor positive allosteric modulator |
Direct Interaction | yes |
CASR | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000036828 | Ensembl Gene Id |
EXTRACELLULAR CALCIUM-SENSING RECEPTOR PRECURSOR (CASR) (PARATHYROID CELL CALCIUM-SENSING RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P41180] | Description |
CASR | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
CASR | Uniprot Gene Name |
ENSG00000036828 | Ensembl Gene Id |
P41180 | Uniprot Accession |
Human Readable Name | DRUGGABLE GENOME |
Interpro Acc | IPR000337 |
Interpro Type | Family |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
CASR | Gene Symbol |
ENSG00000036828 | Ensembl Gene Id |
P41180 | Uniprot Accession |
Target Subclass | GPCR |
Target Subclass | Glutamate |
Target Main Class | Receptors |
CASR | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Glutamate |
ENSG00000036828 | Gene Symbol |
CASR | Ensembl Id |
DRUGGABLE GENOME |
PCAR1 | GENE_SYMBOL |
CASR | GENE_SYMBOL |
Extracellular calcium-sensing receptor | UNIPROT |
PA26097 | PharmGKB ID |
GPRC2A | GO Gene Synonym |
PCAR1 | GO Gene Synonym |
CELL SURFACE, G PROTEIN COUPLED RECEPTOR |
CASR | Gene Symbol |
CLINICALLY ACTIONABLE |
846 | Gene ID |
CAR | dGene Synonym |
EIG8 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
CASR | TTD Gene Abbreviation |
T92076 | TTD Target ID |