1136 |
CHOLINERGIC RECEPTOR NICOTINIC ALPHA 3 SUBUNIT |
CHRNA3 |
LNCR2 |
NACHRA3 |
PAOD2 |
118503 |
1957 |
ENSG00000080644 |
OTTHUMG00000143863 |
P32297 |
ACHA3_HUMAN |
Neuronal acetylcholine receptor subunit alpha-3 |
NEURONAL ACETYLCHOLINE RECEPTOR PROTEIN, ALPHA-3 SUBUNIT PRECURSOR. [SOURCE:UNIPROT/SWISSPROT;ACC:P32297] |
PA113 |
BAIPRCK |
Target Class | Receptors |
Target Subclass | TC:1.A.9 |
Interpro Type | Domain |
Interpro Acc | IPR006202 |
Interpro Name | Neurotransmitter-gated ion-channel |
Human Readable Name | ION CHANNEL |
Uniprot Status | Swiss-Prot |
Interpro Short Name | Neur_chan_lig-bd |
Interpro Acc | IPR006201 |
Interpro Name | Neurotransmitter-gated ion-channel ligand-binding |
Interpro Type | Family |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Neur_channel |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
Direct Interaction | yes |
n/a |
Direct Interaction | yes |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 negative allosteric modulator |
partial agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 partial agonist |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
partial agonist (activating) |
agonist (activating) |
Trial Name | varenicline, CP-526 |
Novel drug target | Established target |
agonist (activating) |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 agonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Mechanism of Interaction | Neuronal acetylcholine receptor; alpha3/beta4 antagonist |
Direct Interaction | yes |
CHRNA3 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
NEURONAL ACETYLCHOLINE RECEPTOR PROTEIN, ALPHA-3 SUBUNIT PRECURSOR. [SOURCE:UNIPROT/SWISSPROT;ACC:P32297] | Description |
CHRNA3 | Display Id |
ENSG00000080644 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
ACHA3_HUMAN | Uniprot Id |
ENSG00000080644 | Ensembl Gene Id |
CHRNA3 | Uniprot Gene Name |
Interpro Acc | IPR006202 |
Interpro Name | Neurotransmitter-gated ion-channel |
Human Readable Name | ION CHANNEL |
ION CHANNEL, DRUGGABLE GENOME |
CHRNA3 | Gene Symbol |
Target Class | Receptors |
Target Subclass | TC:1.A.9 |
PA113 | PharmGKB ID |
ENSG00000080644 | Gene Symbol |
CHRNA3 | Ensembl Id |
DRUGGABLE GENOME |
NACHRA3 | GENE_SYMBOL |
CHRNA3 | GENE_SYMBOL |
Neuronal acetylcholine receptor subunit alpha-3 | UNIPROT |
Neuronal acetylcholine receptor subunit alpha-3 | Gene Name |
P32297 | UniProt ID |
ION CHANNEL |