1588 |
CYTOCHROME P450 FAMILY 19 SUBFAMILY A MEMBER 1 |
CYP19A1 |
ARO |
ARO1 |
CPV1 |
CYAR |
CYP19 |
CYPXIX |
P-450AROM |
107910 |
2594 |
ENSG00000137869 |
OTTHUMG00000131747 |
Cytochrome P450 19A1 |
Aromatase |
Estrogen synthase |
Cytochrome P-450AROM |
P11511 |
CP19A_HUMAN |
PA27091 |
CYTOCHROME P450 19A1 (AROMATASE) (EC 1.14.14.1) (CYPXIX) (ESTROGEN SYNTHETASE) (P-450AROM). [SOURCE:UNIPROT/SWISSPROT;ACC:P11511] |
T13260 |
Target Class | Enzymes |
Target Subclass | EC:1.14.14 |
Human Readable Name | CYTOCHROME P450 |
Interpro Acc | IPR001128 |
Human Readable Name | DRUGGABLE GENOME |
Interpro Name | Cytochrome P450 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Cyt_P450 |
Interpro Type | Family |
Target Main Class | Enzymes |
Transmembrane Helix Count | 2 |
Target Subclass | 1.14.14 |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
CYTOCHROME P450 |
ENZYME |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Cytochrome P450 19A1 inhibitor |
inhibitor (inhibitory) |
Mechanism of Interaction | Cytochrome P450 19A1 inhibitor |
Direct Interaction | yes |
Trial Name | - |
inhibitor (inhibitory) |
Mechanism of Interaction | Cytochrome P450 19A1 inhibitor |
Direct Interaction | yes |
Trial Name | anastrozole,Arimidex |
inhibitor (inhibitory) |
Trial Name | exemestane ,Aromasin |
Novel drug target | Established target |
Mechanism of Interaction | Cytochrome P450 19A1 inhibitor |
inhibitor (inhibitory) |
Notes |
n/a |
Novel drug target | Established target |
Trial Name | atamestane-plus-toremifene |
antagonist (inhibitory) |
inhibitor (inhibitory) |
Trial Name | letrozole ,Femara |
Novel drug target | Established target |
Mechanism of Interaction | Cytochrome P450 19A1 inhibitor |
inhibitor (inhibitory) |
CYP19A1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
CYTOCHROME P450 19A1 (AROMATASE) (EC 1.14.14.1) (CYPXIX) (ESTROGEN SYNTHETASE) (P-450AROM). [SOURCE:UNIPROT/SWISSPROT;ACC:P11511] | Description |
ENSG00000137869 | Ensembl Gene Id |
CYP19A1 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
P11511 | Uniprot Accession |
1588 | Entrez Gene Id |
CYP19A1 | Gene Symbol |
Target Main Class | Enzymes |
Transmembrane Helix Count | 2 |
Target Subclass | 1.14.14 |
1588 | Entrez Gene Id |
ENSG00000137869 | Ensembl Gene Id |
CP19A_HUMAN | Uniprot Id |
Human Readable Name | CYTOCHROME P450 |
Interpro Acc | IPR001128 |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME, CYTOCHROME P450 |
CYP19A1 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:1.14.14 |
PA27091 | PharmGKB ID |
ENSG00000137869 | Gene Symbol |
CYP19A1 | Ensembl Id |
DRUGGABLE GENOME |
AROMATASE | Gene Symbol |
CYAR | GENE_SYMBOL |
CYP19 | GENE_SYMBOL |
CYP19A1 | GENE_SYMBOL |
CYP19A1 | TTD Gene Abbreviation |
T13260 | TTD Target ID |
Aromatase | Gene Name |
P11511 | UniProt ID |
ENZYME |