1723 |
DIHYDROOROTATE DEHYDROGENASE (QUINONE) |
DHODH |
DHOdehase |
POADS |
URA1 |
126064 |
2867 |
ENSG00000102967 |
OTTHUMG00000178093 |
Q02127 |
PYRD_HUMAN |
DIHYDROOROTATE DEHYDROGENASE, MITOCHONDRIAL PRECURSOR (EC 1.3.3.1) (DIHYDROOROTATE OXIDASE) (DHODEHASE). [SOURCE:UNIPROT/SWISSPROT;ACC:Q02127] |
PA27327 |
DIHYDROOROTATE DEHYDROGENASE |
Dihydroorotate oxidase |
Dihydroorotate dehydrogenase (quinone), mitochondrial |
T61400 |
Target Main Class | Enzymes |
Target Subclass | 1.3.3 |
Transmembrane Helix Count | 1 |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Enzymes |
Target Subclass | EC:1.3.3 |
Target Subclass | EC:1.3.5.2 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Type | Conserved_site |
Interpro Name | Dihydroorotate dehydrogenase, conserved site |
Interpro Short Name | Dihydroorotate_DH_CS |
Interpro Acc | IPR001295 |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
inhibitor (inhibitory) |
Mechanism of Interaction | Dihydroorotate dehydrogenase inhibitor |
Direct Interaction | yes |
Trial Name | teriflunomide, HMR1726 |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Dihydroorotate dehydrogenase inhibitor |
Trial Name | - |
inhibitor (inhibitory) |
Trial Name | vidofludimus, 4SC101, SC12267 |
Novel drug target | Established target |
DHODH | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
1723 | Entrez Gene Id |
Q02127 | Uniprot Accession |
DHODH | Gene Symbol |
Target Main Class | Enzymes |
Target Subclass | 1.3.3 |
Transmembrane Helix Count | 1 |
ENSG00000102967 | Ensembl Gene Id |
DIHYDROOROTATE DEHYDROGENASE, MITOCHONDRIAL PRECURSOR (EC 1.3.3.1) (DIHYDROOROTATE OXIDASE) (DHODEHASE). [SOURCE:UNIPROT/SWISSPROT;ACC:Q02127] | Description |
DHODH | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
DHODH | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:1.3.3 |
Target Subclass | EC:1.3.5.2 |
PYRD_HUMAN | Uniprot Id |
DIHYDROOROTATE DEHYDROGENASE (QUINONE), MITOCHONDRIAL | Uniprot Protein Name |
Q02127 | Uniprot Accession |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Type | Conserved_site |
DRUGGABLE GENOME |
PA27327 | PharmGKB ID |
DHODH | GENE_SYMBOL |
Dihydroorotate dehydrogenase (quinone), mitochondrial | UNIPROT |
Dihydroorotate oxidase | UNIPROT |
ENSG00000102967 | Gene Symbol |
DHODH | Ensembl Id |
DRUGGABLE GENOME |
DHODH | TTD Gene Abbreviation |
T61400 | TTD Target ID |