2149 |
COAGULATION FACTOR II THROMBIN RECEPTOR |
F2R |
CF2R |
HTR |
PAR-1 |
PAR1 |
TR |
187930 |
3537 |
ENSG00000181104 |
OTTHUMG00000131299 |
THROMBIN RECEPTOR |
PROTEINASE ACTIVATED RECEPTOR 1 |
COAGULATION FACTOR II RECEPTOR |
P25116 |
PAR1_HUMAN |
PROTEINASE ACTIVATED RECEPTOR 1 PRECURSOR (PAR-1) (THROMBIN RECEPTOR) (COAGULATION FACTOR II RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P25116] |
Proteinase-activated receptor 1 |
T36483 |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Human Readable Name | DRUGGABLE GENOME |
Interpro Type | Family |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000276 |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Uniprot Status | Swiss-Prot |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Proteinase-activated receptor 1 antagonist |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Proteinase-activated receptor 1 antagonist |
antagonist (inhibitory) |
Novel drug target | Novel Target |
Trial Name | vorapaxar , SCH-530348 |
inhibitor (inhibitory) |
Mechanism of Interaction | Proteinase-activated receptor 1 inhibitor |
Direct Interaction | yes |
n/a |
Trial Name | TP-508,Chrysalin |
Novel drug target | Novel Target |
F2R | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
F2R | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
PROTEINASE ACTIVATED RECEPTOR 1 PRECURSOR (PAR-1) (THROMBIN RECEPTOR) (COAGULATION FACTOR II RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P25116] | Description |
ENSG00000181104 | Ensembl Gene Id |
F2R | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PROTEINASE-ACTIVATED RECEPTOR 1 | Uniprot Protein Name |
ENSG00000181104 | Ensembl Gene Id |
P25116 | Uniprot Accession |
Interpro Type | Family |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000276 |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
ENSG00000181104 | Gene Symbol |
F2R | Ensembl Id |
DRUGGABLE GENOME |
PAR1 | GENE_SYMBOL |
TR | GENE_SYMBOL |
F2R | GENE_SYMBOL |
CF2R | GO Gene Synonym |
PAR1 | GO Gene Synonym |
TR | GO Gene Synonym |
CELL SURFACE, G PROTEIN COUPLED RECEPTOR |
2149 | Gene ID |
CF2R | dGene Synonym |
HTR | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
F2R | TTD Gene Abbreviation |
T36483 | TTD Target ID |