9568 |
GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR SUBUNIT 2 |
GABBR2 |
GABABR2 |
GPR51 |
GPRC3B |
HG20 |
HRIHFB2099 |
607340 |
4507 |
ENSG00000136928 |
OTTHUMG00000020345 |
G-protein coupled receptor 51 |
GABA-B receptor 2 |
GABA-B-R2 |
GABA-BR2 |
Gb2 |
GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR, SUBUNIT 2 PRECURSOR (GABA-B RECEPTOR 2) (GABA-B-R2) (GB2) (GABABR2) (G-PROTEIN COUPLED RECEPTOR 51) (GPR 51) (HG20). [SOURCE:UNIPROT/SWISSPROT;ACC:O75899] |
O75899 |
GABR2_HUMAN |
DEE59 |
EIEE59 |
NDPLHS |
Human Readable Name | DRUGGABLE GENOME |
Target Subclass | Glutamate |
Transmembrane Helix Count | 7 |
Target Subclass | GPCR |
Target Main Class | Receptors |
Target Class | Receptors |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Short Name | GPCR_3 |
Interpro Type | Family |
Interpro Name | GPCR, family 3 |
Interpro Acc | IPR000337 |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
agonist (activating) |
Trial Name | Arbaclofen |
Novel drug target | Established target |
Direct Interaction | yes |
agonist (activating) |
Trial Name | ALKS 29 |
Novel drug target | Established target |
Mechanism of Interaction | GABA-B receptor agonist |
agonist (activating) |
Mechanism of Interaction | GABA-B receptor 2 agonist |
Direct Interaction | yes |
Trial Name | lesogaberan, AZD-3355 |
agonist (activating) |
Mechanism of Interaction | GABA-B receptor agonist |
Direct Interaction | yes |
GABBR2 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000136928 | Ensembl Gene Id |
9568 | Entrez Gene Id |
GABBR2 | Gene Symbol |
Target Subclass | Glutamate |
Transmembrane Helix Count | 7 |
Target Subclass | GPCR |
GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR SUBUNIT 2 | Uniprot Protein Name |
GABR2_HUMAN | Uniprot Id |
O75899 | Uniprot Accession |
Interpro Type | Family |
Interpro Name | GPCR, family 3 |
Interpro Acc | IPR000337 |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
GPR51 | Display Id |
GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR, SUBUNIT 2 PRECURSOR (GABA-B RECEPTOR 2) (GABA-B-R2) (GB2) (GABABR2) (G-PROTEIN COUPLED RECEPTOR 51) (GPR 51) (HG20). [SOURCE:UNIPROT/SWISSPROT;ACC:O75899] | Description |
ENSG00000136928 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
GABBR2 | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Glutamate |
ENSG00000136928 | Gene Symbol |
GABBR2 | Ensembl Id |
DRUGGABLE GENOME |
GPRC3B | GENE_SYMBOL |
GABBR2 | GENE_SYMBOL |
Gamma-aminobutyric acid type B receptor subunit 2 | UNIPROT |
9568 | Gene ID |
GABABR2 | dGene Synonym |
GPR51 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
Gamma-aminobutyric acid type B receptor subunit 2 | Gene Name |
O75899 | UniProt ID |
ION CHANNEL |