2898 |
GLUTAMATE IONOTROPIC RECEPTOR KAINATE TYPE SUBUNIT 2 |
GRIK2 |
EAA4 |
GLR6 |
GLUK6 |
GLUR6 |
GluK2 |
MRT6 |
138244 |
4580 |
ENSG00000164418 |
OTTHUMG00000016328 |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 2 PRECURSOR (GLUTAMATE RECEPTOR 6) (GLUR-6) (GLUR6) (EXCITATORY AMINO ACID RECEPTOR 4) (EAA4). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13002] |
Q13002 |
GRIK2_HUMAN |
KA2 |
EAA2 |
GRIK5 |
Glutamate receptor ionotropic, kainate 5 |
Excitatory amino acid receptor 2 |
Glutamate receptor KA-2 |
GluK5 |
GluR-6 |
Glutamate receptor 6 |
Excitatory amino acid receptor 4 |
Glutamate receptor ionotropic, kainate 2 |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 2 |
NEDLAS |
Human Readable Name | DRUGGABLE GENOME |
Target Subclass | Glutamate |
Target Subclass | Ligand_gated_ion_channels |
Target Subclass | Channels |
Transmembrane Helix Count | 3 |
Target Main Class | Receptors |
Interpro Acc | IPR001320 |
Interpro Short Name | Iontro_glu_rcpt |
Interpro Type | Domain |
Interpro Name | Ionotropic glutamate receptor |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Target Class | Receptors |
Target Subclass | TC:1.A.10.1 |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
Direct Interaction | yes |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
antagonist (inhibitory) |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | - |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
GRIK2 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 2 | Uniprot Protein Name |
GRIK2 | Uniprot Gene Name |
ENSG00000164418 | Ensembl Gene Id |
Interpro Acc | IPR001320 |
Interpro Short Name | Iontro_glu_rcpt |
Interpro Type | Domain |
DRUGGABLE GENOME |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 2 PRECURSOR (GLUTAMATE RECEPTOR 6) (GLUR-6) (GLUR6) (EXCITATORY AMINO ACID RECEPTOR 4) (EAA4). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13002] | Description |
GRIK2 | Display Id |
ENSG00000164418 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
GRIK2 | Gene Symbol |
GRIK2_HUMAN | Uniprot Id |
Q13002 | Uniprot Accession |
Target Subclass | Glutamate |
Target Subclass | Ligand_gated_ion_channels |
Target Subclass | Channels |
GRIK2 | Gene Symbol |
Target Class | Receptors |
Target Subclass | TC:1.A.10.1 |
GLUR6 | GENE_SYMBOL |
GRIK2 | GENE_SYMBOL |
Glutamate receptor ionotropic, kainate 2 | UNIPROT |
ENSG00000164418 | Gene Symbol |
GRIK2 | Ensembl Id |
DRUGGABLE GENOME |
GRIK2 | GENE_SYMBOL |
GRIK5 | GENE_SYMBOL |
Glutamate receptor ionotropic, kainate 5 | UNIPROT |
Glutamate receptor ionotropic, kainate 2 | Gene Name |
Q13002 | UniProt ID |
ION CHANNEL |