2899 |
GLUTAMATE IONOTROPIC RECEPTOR KAINATE TYPE SUBUNIT 3 |
GRIK3 |
EAA5 |
GLR7 |
GLUR7 |
GluK3 |
GluR7a |
138243 |
4581 |
ENSG00000163873 |
OTTHUMG00000004189 |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 3 PRECURSOR (GLUTAMATE RECEPTOR 7) (GLUR-7) (GLUR7) (EXCITATORY AMINO ACID RECEPTOR 5) (EAA5). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13003] |
Q13003 |
Excitatory amino acid receptor 5 |
Glutamate receptor ionotropic, kainate 3 |
Glutamate receptor 7 |
GluR-7 |
GRIK3_HUMAN |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 3 |
PA28975 |
Human Readable Name | DRUGGABLE GENOME |
Interpro Acc | IPR001320 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Type | Domain |
Interpro Short Name | Iontro_glu_rcpt |
Interpro Name | Ionotropic glutamate receptor |
Target Class | Receptors |
Target Subclass | TC:1.A.10.1 |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
antagonist (inhibitory) |
Novel drug target | Novel Target |
Trial Name | tezampanel, NGX424,NGX426 |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
antagonist (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
antagonist (inhibitory) |
Mechanism of Interaction | Glutamate receptor ionotropic kainate antagonist |
Direct Interaction | yes |
GRIK3 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
Q13003 | Uniprot Accession |
GRIK3_HUMAN | Uniprot Id |
ENSG00000163873 | Ensembl Gene Id |
Interpro Acc | IPR001320 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
DRUGGABLE GENOME |
GRIK3 | Gene Symbol |
Target Class | Receptors |
Target Subclass | TC:1.A.10.1 |
GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 3 PRECURSOR (GLUTAMATE RECEPTOR 7) (GLUR-7) (GLUR7) (EXCITATORY AMINO ACID RECEPTOR 5) (EAA5). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13003] | Description |
GRIK3 | Display Id |
ENSG00000163873 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PA28975 | PharmGKB ID |
ENSG00000163873 | Gene Symbol |
GRIK3 | Ensembl Id |
DRUGGABLE GENOME |
GLUR7 | GENE_SYMBOL |
GRIK3 | GENE_SYMBOL |
Glutamate receptor ionotropic, kainate 3 | UNIPROT |
Glutamate receptor ionotropic, kainate 3 | Gene Name |
Q13003 | UniProt ID |
ION CHANNEL |