• GRIK5 2901 Druggable Genome

    Alternate Names:

    2901
    GLUTAMATE IONOTROPIC RECEPTOR KAINATE TYPE SUBUNIT 5
    GRIK5
    EAA2
    GRIK2
    GluK5
    KA2
    600283
    4583
    ENSG00000105737
    OTTHUMG00000044573
    GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 5 PRECURSOR (GLUTAMATE RECEPTOR KA-2) (KA2) (EXCITATORY AMINO ACID RECEPTOR 2) (EAA2). [SOURCE:UNIPROT/SWISSPROT;ACC:Q16478]
    Q16478
    GRIK5_HUMAN
    GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 5
    Glutamate receptor ionotropic, kainate 5

    Gene Info:

    Human Readable Name DRUGGABLE GENOME
    Uniprot Evidence 2: Evidence at transcript level
    Interpro Acc IPR001320
    Uniprot Status Swiss-Prot
    Interpro Type Domain
    Interpro Short Name Iontro_glu_rcpt
    Interpro Name Ionotropic glutamate receptor
    Target Class Receptors
    Target Subclass TC:1.A.10.1
    Gene Biotype PROTEIN_CODING
    (2 More Sources)

    Gene Categories: Category Details

    ION CHANNEL
    DRUGGABLE GENOME

    Publications:

  • Interaction Score: 6.87

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Trial Name tezampanel, NGX424,NGX426
    Novel drug target Novel Target

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

    • Version: 101_38

    Alternate Names:
    GRIK5 Ensembl Gene Name

    Gene Info:
    Gene Biotype PROTEIN_CODING

    Publications:

    • Version: 26-July-2011

    Alternate Names:
    GRIK5 Display Id
    ENSG00000105737 Ensembl Gene Id
    GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 5 PRECURSOR (GLUTAMATE RECEPTOR KA-2) (KA2) (EXCITATORY AMINO ACID RECEPTOR 2) (EAA2). [SOURCE:UNIPROT/SWISSPROT;ACC:Q16478] Description

    Gene Info:
    Human Readable Name DRUGGABLE GENOME

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: 11-September-2012

    Alternate Names:
    GRIK5 Uniprot Gene Name
    GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 5 Uniprot Protein Name
    2901 Entrez Gene Id

    Gene Info:
    Uniprot Evidence 2: Evidence at transcript level
    Interpro Acc IPR001320
    Uniprot Status Swiss-Prot

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: January-2014

    Alternate Names:
    GRIK5 Gene Symbol

    Gene Info:
    Target Class Receptors
    Target Subclass TC:1.A.10.1

    Publications:

    • Version: 31-May-2017

    Alternate Names:
    ENSG00000105737 Gene Symbol
    GRIK5 Ensembl Id

    Gene Info:

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: 01-February-2022

    Alternate Names:
    Glutamate receptor ionotropic, kainate 5 Gene Name
    Q16478 UniProt ID

    Gene Info:

    Gene Categories:
    ION CHANNEL

    Publications: