3363 |
5-HYDROXYTRYPTAMINE RECEPTOR 7 |
HTR7 |
5-HT7 |
182137 |
5302 |
ENSG00000148680 |
OTTHUMG00000018732 |
P34969 |
5HT7R_HUMAN |
5-HT-7 |
Serotonin receptor 7 |
5-HT-X |
5-HYDROXYTRYPTAMINE 7 RECEPTOR (5-HT-7) (SEROTONIN RECEPTOR 7) (5-HT- X) (5HT7). [SOURCE:UNIPROT/SWISSPROT;ACC:P34969] |
PA29561 |
5-HT 7 receptor |
T79062 |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Interpro Acc | IPR000276 |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | DRUGGABLE GENOME |
Interpro Type | Family |
Uniprot Status | Swiss-Prot |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
Gene Biotype | PROTEIN_CODING |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
antagonist (inhibitory) |
antagonist (inhibitory) |
Mechanism of Interaction | Serotonin 7 (5-HT7) receptor antagonist |
Direct Interaction | yes |
antagonist (inhibitory) |
Trial Name | lurasidone, SM-13496,Latuda |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | Lu AA21004 |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
n/a |
Trial Name | OPC-34712 |
Novel drug target | Established target |
n/a |
Trial Name | bifeprunox, DU127090 |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | Asenapine |
Novel drug target | Established target |
n/a |
Trial Name | pardoprunox, SLV 308 |
Novel drug target | Established target |
antagonist (inhibitory) |
Novel drug target | Established target |
Trial Name | iloperidone,Fanapt, Fiapta, Zomaril |
antagonist (inhibitory) |
Trial Name | ALKS 3831 |
Trial Name | OREX-003, olanzapine plus zonisamide SR |
Trial Name | Olanzapine/fluoxetine combination,Symbyax (Zyprexa/Prozac) |
HTR7 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000148680 | Ensembl Gene Id |
5HT7R_HUMAN | Uniprot Id |
P34969 | Uniprot Accession |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Interpro Acc | IPR000276 |
Uniprot Evidence | 1: Evidence at protein level |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
HTR7 | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
P34969 | Uniprot Accession |
HTR7 | Gene Symbol |
3363 | Entrez Gene Id |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
Target Subclass | Rhodopsin |
5-HYDROXYTRYPTAMINE 7 RECEPTOR (5-HT-7) (SEROTONIN RECEPTOR 7) (5-HT- X) (5HT7). [SOURCE:UNIPROT/SWISSPROT;ACC:P34969] | Description |
ENSG00000148680 | Ensembl Gene Id |
HTR7 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PA29561 | PharmGKB ID |
ENSG00000148680 | Gene Symbol |
HTR7 | Ensembl Id |
DRUGGABLE GENOME |
HTR7 | GENE_SYMBOL |
5-hydroxytryptamine receptor 7 | UNIPROT |
5-HT-X | UNIPROT |
3363 | Gene ID |
5-HT7 | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
HTR7 | TTD Gene Abbreviation |
T79062 | TTD Target ID |