3615 |
INOSINE MONOPHOSPHATE DEHYDROGENASE 2 |
IMPDH2 |
IMPD2 |
IMPDH-II |
146691 |
6053 |
ENSG00000178035 |
OTTHUMG00000156771 |
PA29863 |
P12268 |
IMPD 2 |
Inosine-5'-monophosphate dehydrogenase 2 |
IMP dehydrogenase 2 |
IMPDH 2 |
IMDH2_HUMAN |
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 2 (EC 1.1.1.205) (IMP DEHYDROGENASE 2) (IMPDH-II) (IMPD 2). [SOURCE:UNIPROT/SWISSPROT;ACC:P12268] |
T89360 |
Target Main Class | Enzymes |
Target Subclass | 1.1.1.205 |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | IMP_DH_GMPRt |
Interpro Acc | IPR001093 |
Interpro Name | IMP dehydrogenase/GMP reductase |
Uniprot Status | Swiss-Prot |
Interpro Type | Domain |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Enzymes |
Target Subclass | EC:1.1.1.205 |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
ENZYME |
inhibitor (inhibitory) |
Mechanism of Interaction | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor |
Direct Interaction | yes |
n/a |
Trial Name | AVN-944 |
Novel drug target | Established target |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor |
inhibitor (inhibitory) |
Mechanism of Interaction | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor |
Direct Interaction | yes |
IMPDH2 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000178035 | Ensembl Gene Id |
IMDH2_HUMAN | Uniprot Id |
3615 | Entrez Gene Id |
Target Main Class | Enzymes |
Target Subclass | 1.1.1.205 |
P12268 | Uniprot Accession |
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 2 | Uniprot Protein Name |
IMPDH2 | Uniprot Gene Name |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | IMP_DH_GMPRt |
Interpro Acc | IPR001093 |
DRUGGABLE GENOME |
ENSG00000178035 | Ensembl Gene Id |
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 2 (EC 1.1.1.205) (IMP DEHYDROGENASE 2) (IMPDH-II) (IMPD 2). [SOURCE:UNIPROT/SWISSPROT;ACC:P12268] | Description |
IMPDH2 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
IMPDH2 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:1.1.1.205 |
PA29863 | PharmGKB ID |
ENSG00000178035 | Gene Symbol |
IMPDH2 | Ensembl Id |
DRUGGABLE GENOME |
IMPD2 | GENE_SYMBOL |
IMPDH2 | GENE_SYMBOL |
Inosine-5'-monophosphate dehydrogenase 2 | UNIPROT |
IMPDH2 | TTD Gene Abbreviation |
T89360 | TTD Target ID |
Inosine-5'-monophosphate dehydrogenase 2 | Gene Name |
P12268 | UniProt ID |
ENZYME |