• Interaction Score: 15.9

    Interaction Types & Directionality:
    activator (activating)
    blocker (inhibitory)

    Interaction Info:
    Trial Name retigabine, ezogabine,Potiga
    Novel drug target Established target
    Mechanism of Interaction KCNQ (Kv7) potassium channel blocker

  • Interaction Score: 1.77

    Interaction Types & Directionality:
    activator (activating)

    Interaction Info:
    Mechanism of Interaction Voltage-gated potassium channel subunit Kv7.2 activator
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.28

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    22336956


    Sources:
    PharmGKB

  • Interaction Score: 0.23

    Interaction Types & Directionality:
    blocker (inhibitory)

    Interaction Info:
    Mechanism of Interaction Voltage-gated potassium channel blocker
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.23

    Interaction Types & Directionality:
    blocker (inhibitory)

    Interaction Info:
    Mechanism of Interaction Voltage-gated potassium channel blocker
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.21

    Interaction Types & Directionality:
    blocker (inhibitory)

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction Voltage-gated potassium channel blocker

    PMIDs:
    None found


  • Interaction Score: 0.18

    Interaction Types & Directionality:
    blocker (inhibitory)

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction Voltage-gated potassium channel blocker

    PMIDs:
    None found