5607 |
MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 |
MAP2K5 |
HsT17454 |
MAPKK5 |
MEK5 |
PRKMK5 |
602520 |
6845 |
ENSG00000137764 |
OTTHUMG00000133264 |
Q13163 |
MP2K5_HUMAN |
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 |
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 (EC 2.7.1.-) (MAP KINASE KINASE 5) (MAPKK 5) (MAPK/ERK KINASE 5). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13163] |
MKK5 |
Interpro Acc | IPR002290 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Ser/Thr_dual-sp_kinase_dom |
Interpro Name | Serine/threonine- / dual-specificity protein kinase, catalytic domain |
Interpro Type | Domain |
Human Readable Name | DRUGGABLE GENOME |
Human Readable Name | KINASE |
Target Class | Enzymes |
Target Subclass | EC:2.7.12.2 |
Gene Biotype | PROTEIN_CODING |
KINASE |
SERINE THREONINE KINASE |
TYROSINE KINASE |
DRUGGABLE GENOME |
n/a |
Novel drug target | Novel Target |
Trial Name | WX-554 |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
inhibitor (inhibitory) |
MAP2K5 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 (EC 2.7.1.-) (MAP KINASE KINASE 5) (MAPKK 5) (MAPK/ERK KINASE 5). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13163] | Description |
MAP2K5 | Display Id |
ENSG00000137764 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 5 | Uniprot Protein Name |
MP2K5_HUMAN | Uniprot Id |
MAP2K5 | Uniprot Gene Name |
Interpro Acc | IPR002290 |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
KINASE, DRUGGABLE GENOME |
MAP2K5 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:2.7.12.2 |
ENSG00000137764 | Gene Symbol |
MAP2K5 | Ensembl Id |
DRUGGABLE GENOME |
MEK5 | GO Gene Synonym |
MKK5 | GO Gene Synonym |
PRKMK5 | GO Gene Synonym |
SERINE THREONINE KINASE, TYROSINE KINASE |
5607 | Gene ID |
HsT17454 | dGene Synonym |
MAPKK5 | dGene Synonym |
KINASE, SERINE THREONINE KINASE |
Dual specificity mitogen-activated protein kinase kinase 5 | Gene Name |
Q13163 | UniProt ID |
KINASE |