6300 |
MITOGEN-ACTIVATED PROTEIN KINASE 12 |
MAPK12 |
ERK-6 |
ERK3 |
ERK6 |
MAPK 12 |
P38GAMMA |
PRKM12 |
SAPK-3 |
SAPK3 |
602399 |
6874 |
ENSG00000188130 |
OTTHUMG00000030145 |
P53778 |
MK12_HUMAN |
MITOGEN-ACTIVATED PROTEIN KINASE 12 (EC 2.7.1.37) (EXTRACELLULAR SIGNAL-REGULATED KINASE 6) (ERK-6) (ERK5) (STRESS-ACTIVATED PROTEIN KINASE-3) (MITOGEN-ACTIVATED PROTEIN KINASE P38 GAMMA) (MAP KINASE P38 GAMMA). [SOURCE:UNIPROT/SWISSPROT;ACC:P53778] |
PA30619 |
MAP KINASE P38 |
T79798 |
Interpro Acc | IPR002290 |
Interpro Name | Serine/threonine- / dual-specificity protein kinase, catalytic domain |
Interpro Type | Domain |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | Ser/Thr_dual-sp_kinase_dom |
Human Readable Name | KINASE |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Status | Swiss-Prot |
Target Class | Enzymes |
Target Subclass | EC:2.7.11.24 |
Gene Biotype | PROTEIN_CODING |
TUMOR SUPPRESSOR |
KINASE |
SERINE THREONINE KINASE |
DRUGGABLE GENOME |
ENZYME |
TRANSCRIPTION FACTOR |
n/a |
Trial Name | ARRY-797 |
Novel drug target | Novel Target |
n/a |
Trial Name | PH-797804 |
Novel drug target | Novel Target |
n/a |
Trial Name | BMS-582949 |
Novel drug target | Novel Target |
n/a |
Novel drug target | Novel Target |
Trial Name | CPSI-2364 |
n/a |
Trial Name | ARRY-614 |
Novel drug target | Novel Target |
n/a |
Trial Name | VX-702 |
Novel drug target | Novel Target |
n/a |
Trial Name | pirfenidone,Esbriet , Deskar, Pirespa |
Novel drug target | Novel Target |
inhibitor (inhibitory) |
MAPK12 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
MAPK12 | Uniprot Gene Name |
6300 | Entrez Gene Id |
MK12_HUMAN | Uniprot Id |
Interpro Acc | IPR002290 |
Interpro Name | Serine/threonine- / dual-specificity protein kinase, catalytic domain |
Interpro Type | Domain |
KINASE, DRUGGABLE GENOME |
MAPK12 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:2.7.11.24 |
MAPK12 | Display Id |
MITOGEN-ACTIVATED PROTEIN KINASE 12 (EC 2.7.1.37) (EXTRACELLULAR SIGNAL-REGULATED KINASE 6) (ERK-6) (ERK5) (STRESS-ACTIVATED PROTEIN KINASE-3) (MITOGEN-ACTIVATED PROTEIN KINASE P38 GAMMA) (MAP KINASE P38 GAMMA). [SOURCE:UNIPROT/SWISSPROT;ACC:P53778] | Description |
ENSG00000188130 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PA30619 | PharmGKB ID |
ENSG00000188130 | Gene Symbol |
MAPK12 | Ensembl Id |
DRUGGABLE GENOME |
ENSG00000188130 | Ensembl Gene ID |
ERK6 | Human Protein Atlas Gene Synonym |
p38gamma | Human Protein Atlas Gene Synonym |
ENZYME |
ERK6 | GO Gene Synonym |
SAPK3 | GO Gene Synonym |
TUMOR SUPPRESSOR, SERINE THREONINE KINASE |
6300 | Gene ID |
ERK3 | dGene Synonym |
ERK6 | dGene Synonym |
KINASE, SERINE THREONINE KINASE |
MAPK12 | TTD Gene Abbreviation |
T79798 | TTD Target ID |
Mitogen-activated protein kinase 12 | Gene Name |
P53778 | UniProt ID |
KINASE, TRANSCRIPTION FACTOR |