5599 |
MITOGEN-ACTIVATED PROTEIN KINASE 8 |
MAPK8 |
JNK |
JNK-46 |
JNK1 |
JNK1A2 |
JNK21B1/2 |
PRKM8 |
SAPK1 |
SAPK1c |
601158 |
6881 |
ENSG00000107643 |
OTTHUMG00000018172 |
P45983 |
PA283 |
MAPK 8 |
MAP kinase 8 |
c-Jun N-terminal kinase 1 |
Stress-activated protein kinase JNK1 |
Stress-activated protein kinase 1c |
MK08_HUMAN |
MITOGEN-ACTIVATED PROTEIN KINASE 8 (EC 2.7.1.37) (STRESS-ACTIVATED PROTEIN KINASE JNK1) (C-JUN N-TERMINAL KINASE 1) (JNK-46). [SOURCE:UNIPROT/SWISSPROT;ACC:P45983] |
T40097 |
Jun N terminal kinase |
T85421 |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Enzymes |
Target Subclass | EC:2.7.11.24 |
Interpro Type | Domain |
Human Readable Name | KINASE |
Interpro Short Name | Ser/Thr_dual-sp_kinase_dom |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Name | Serine/threonine- / dual-specificity protein kinase, catalytic domain |
Uniprot Status | Swiss-Prot |
Interpro Acc | IPR002290 |
Gene Biotype | PROTEIN_CODING |
KINASE |
SERINE THREONINE KINASE |
DRUGGABLE GENOME |
TRANSCRIPTION FACTOR |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | c-Jun N-terminal kinase 1 inhibitor |
n/a |
Trial Name | AM-111 |
Novel drug target | Novel Target |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | c-Jun N-terminal kinase 1 inhibitor |
inhibitor (inhibitory) |
Mechanism of Interaction | c-Jun N-terminal kinase, JNK inhibitor |
Direct Interaction | yes |
MAPK8 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
MITOGEN-ACTIVATED PROTEIN KINASE 8 (EC 2.7.1.37) (STRESS-ACTIVATED PROTEIN KINASE JNK1) (C-JUN N-TERMINAL KINASE 1) (JNK-46). [SOURCE:UNIPROT/SWISSPROT;ACC:P45983] | Description |
ENSG00000107643 | Ensembl Gene Id |
MAPK8 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
MAPK8 | Uniprot Gene Name |
MK08_HUMAN | Uniprot Id |
ENSG00000107643 | Ensembl Gene Id |
Interpro Type | Domain |
Human Readable Name | KINASE |
Interpro Short Name | Ser/Thr_dual-sp_kinase_dom |
KINASE, DRUGGABLE GENOME |
MAPK8 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:2.7.11.24 |
PA283 | PharmGKB ID |
ENSG00000107643 | Gene Symbol |
MAPK8 | Ensembl Id |
DRUGGABLE GENOME |
PRKM8 | GENE_SYMBOL |
SAPK1 | GENE_SYMBOL |
SAPK1C | GENE_SYMBOL |
JNK1 | GO Gene Synonym |
PRKM8 | GO Gene Synonym |
SAPK1 | GO Gene Synonym |
SERINE THREONINE KINASE |
5599 | Gene ID |
JNK | dGene Synonym |
JNK-46 | dGene Synonym |
KINASE, SERINE THREONINE KINASE |
JNK | TTD Gene Abbreviation |
T85421 | TTD Target ID |
JNK1 | TTD Gene Abbreviation |
T40097 | TTD Target ID |
Mitogen-activated protein kinase 8 | Gene Name |
P45983 | UniProt ID |
KINASE, TRANSCRIPTION FACTOR |