4486 |
MACROPHAGE STIMULATING 1 RECEPTOR |
MST1R |
CD136 |
CDw136 |
NPCA3 |
PTK8 |
RON |
600168 |
7381 |
ENSG00000164078 |
OTTHUMG00000156709 |
Macrophage-stimulating protein receptor alpha chain |
p185-Ron |
MSP receptor |
CD_antigen=CD136 |
Macrophage-stimulating protein receptor |
Protein-tyrosine kinase 8 |
Macrophage-stimulating protein receptor beta chain |
MACROPHAGE-STIMULATING PROTEIN RECEPTOR PRECURSOR (EC 2.7.1.112) (MSP RECEPTOR) (P185-RON) (CDW136) (CD136 ANTIGEN). [SOURCE:UNIPROT/SWISSPROT;ACC:Q04912] |
Q04912 |
RON_HUMAN |
T01973 |
SEA |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Enzymes |
Target Subclass | EC:2.7.10.1 |
Human Readable Name | KINASE |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR001245 |
Interpro Name | Serine-threonine/tyrosine-protein kinase catalytic domain |
Interpro Type | Domain |
Interpro Short Name | Ser-Thr/Tyr_kinase_cat_dom |
Uniprot Status | Swiss-Prot |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
KINASE |
TYROSINE KINASE |
DRUGGABLE GENOME |
CLINICALLY ACTIONABLE |
ENZYME |
inhibitor (inhibitory) |
Mechanism of Interaction | Macrophage-stimulating protein receptor inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Notes | |
Trial Name | MGCD265 |
Novel drug target | Novel Target |
inhibitor (inhibitory) |
Mechanism of Interaction | Macrophage-stimulating protein receptor inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Notes |
inhibitor (inhibitory) |
MST1R | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
MST1R | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:2.7.10.1 |
MACROPHAGE-STIMULATING PROTEIN RECEPTOR PRECURSOR (EC 2.7.1.112) (MSP RECEPTOR) (P185-RON) (CDW136) (CD136 ANTIGEN). [SOURCE:UNIPROT/SWISSPROT;ACC:Q04912] | Description |
ENSG00000164078 | Ensembl Gene Id |
MST1R | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
RON_HUMAN | Uniprot Id |
4486 | Entrez Gene Id |
MACROPHAGE-STIMULATING PROTEIN RECEPTOR ALPHA CHAIN | Uniprot Protein Name |
Human Readable Name | KINASE |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR001245 |
KINASE, DRUGGABLE GENOME |
RON | Gene Symbol |
ENSG00000164078 | Gene Symbol |
MST1R | Ensembl Id |
DRUGGABLE GENOME |
RON | GENE_SYMBOL |
MST1R | GENE_SYMBOL |
Macrophage-stimulating protein receptor | UNIPROT |
ENSG00000164078 | Ensembl Gene ID |
CD136 | Human Protein Atlas Gene Synonym |
CDw136 | Human Protein Atlas Gene Synonym |
CELL SURFACE, ENZYME |
PTK8 | GO Gene Synonym |
RON | GO Gene Synonym |
CELL SURFACE |
4486 | Gene ID |
CD136 | dGene Synonym |
CDw136 | dGene Synonym |
KINASE, TYROSINE KINASE |
RON | TTD Gene Abbreviation |
T01973 | TTD Target ID |
Macrophage-stimulating protein receptor | Gene Name |
Q04912 | UniProt ID |
KINASE |
CLINICALLY ACTIONABLE |