4881 |
NATRIURETIC PEPTIDE RECEPTOR 1 |
NPR1 |
ANPRA |
ANPa |
GUC2A |
GUCY2A |
NPRA |
108960 |
7943 |
ENSG00000169418 |
OTTHUMG00000037085 |
P16066 |
ATRIAL NATRIURETIC PEPTIDE RECEPTOR 1 |
ANPRA_HUMAN |
ANP-A |
NPR-A |
ANPR-A |
Guanylate cyclase A |
Atrial natriuretic peptide receptor type A |
GC-A |
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A |
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A PRECURSOR (ANP-A) (ANPRA) (GC-A) (GUANYLATE CYCLASE) (EC 4.6.1.2) (NPR-A) (ATRIAL NATRIURETIC PEPTIDE A-TYPE RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P16066] |
T71230 |
Interpro Acc | IPR001245 |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Interpro Type | Family |
Interpro Type | Domain |
Interpro Acc | IPR001170 |
Interpro Short Name | Ntpep_rcpt |
Human Readable Name | DRUGGABLE GENOME |
Interpro Short Name | A/G_cyclase |
Interpro Name | Natriuretic peptide receptor |
Interpro Acc | IPR001054 |
Interpro Short Name | Ser-Thr/Tyr_kinase_cat_dom |
Human Readable Name | KINASE |
Interpro Name | Serine-threonine/tyrosine-protein kinase catalytic domain |
Interpro Name | Adenylyl cyclase class-3/4/guanylyl cyclase |
Target Subclass | RGC |
Target Main Class | Receptors |
Transmembrane Helix Count | 1 |
Target Subclass | Kinase |
Target Class | Receptors |
Target Subclass | EC:4.6.1.2 |
Gene Biotype | PROTEIN_CODING |
KINASE |
DRUGGABLE GENOME |
agonist (activating) |
Trial Name | PL-3994 |
Novel drug target | Established target |
agonist (activating) |
Trial Name | - |
Novel drug target | Established target |
agonist (activating) |
binder |
Mechanism of Interaction | Atrial natriuretic peptide receptor A agonist |
Direct Interaction | yes |
Trial Name | nesiritide ,Natrecor |
agonist (activating) |
n/a |
Trial Name | - |
Novel drug target | Established target |
agonist (activating) |
Trial Name | MQX-503, nitroglycerin 0.9% topical cream,Vascana |
Novel drug target | Established target |
NPR1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A PRECURSOR (ANP-A) (ANPRA) (GC-A) (GUANYLATE CYCLASE) (EC 4.6.1.2) (NPR-A) (ATRIAL NATRIURETIC PEPTIDE A-TYPE RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P16066] | Description |
NPR1 | Display Id |
ENSG00000169418 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
NPR1 | Gene Symbol |
Target Class | Receptors |
Target Subclass | EC:4.6.1.2 |
NPR1 | Gene Symbol |
P16066 | Uniprot Accession |
ANPRA_HUMAN | Uniprot Id |
Target Subclass | RGC |
Target Main Class | Receptors |
Transmembrane Helix Count | 1 |
ANPRA_HUMAN | Uniprot Id |
ATRIAL NATRIURETIC PEPTIDE RECEPTOR 1 | Uniprot Protein Name |
4881 | Entrez Gene Id |
Interpro Acc | IPR001245 |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
KINASE, DRUGGABLE GENOME |
NPR1 | TTD Gene Abbreviation |
T71230 | TTD Target ID |
ENSG00000169418 | Gene Symbol |
NPR1 | Ensembl Id |
DRUGGABLE GENOME |
ANPRA | GENE_SYMBOL |
NPR1 | GENE_SYMBOL |
Atrial natriuretic peptide receptor 1 | UNIPROT |
Atrial natriuretic peptide receptor 1 | Gene Name |
P16066 | UniProt ID |
KINASE |