• PLA2G10 8399 Druggable Genome

    Alternate Names:

    8399
    PHOSPHOLIPASE A2 GROUP X
    PLA2G10
    GXPLA2
    GXSPLA2
    SPLA2
    sPLA2-X
    603603
    9029
    ENSG00000069764
    OTTHUMG00000048069
    GROUP X SECRETORY PHOSPHOLIPASE A2 PRECURSOR (EC 3.1.1.4) (PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX) (GX SPLA2) (SPLA2-X). [SOURCE:UNIPROT/SWISSPROT;ACC:O15496]
    O15496
    PA2GX_HUMAN
    GX sPLA2
    Phosphatidylcholine 2-acylhydrolase 10
    Group X secretory phospholipase A2
    Group 10 secretory phospholipase A2

    Gene Info:

    Human Readable Name DRUGGABLE GENOME
    Target Class Enzymes
    Target Subclass EC:3.1.1.4
    Uniprot Status Swiss-Prot
    Interpro Short Name PLipase_A2_euk
    Interpro Type Family
    Human Readable Name PHOSPHOLIPASE
    Interpro Name Phospholipase A2, eukaryotic
    Interpro Acc IPR001211
    Uniprot Evidence 1: Evidence at protein level
    Gene Biotype PROTEIN_CODING
    (4 More Sources)

    Gene Categories: Category Details

    PHOSPHOLIPASE
    DRUGGABLE GENOME
    ENZYME

    Publications:

  • Interaction Score: 10.3

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Group X secretory phospholipase A2 inhibitor
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 10.3

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Trial Name varespladib, A-002
    Novel drug target Novel Target
    Trial Name varespladib sodium, A-001

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

    • Version: 101_38

    Alternate Names:
    PLA2G10 Ensembl Gene Name

    Gene Info:
    Gene Biotype PROTEIN_CODING

    Publications:

    • Version: 26-July-2011

    Alternate Names:
    ENSG00000069764 Ensembl Gene Id
    PLA2G10 Display Id
    GROUP X SECRETORY PHOSPHOLIPASE A2 PRECURSOR (EC 3.1.1.4) (PHOSPHATIDYLCHOLINE 2-ACYLHYDROLASE GX) (GX SPLA2) (SPLA2-X). [SOURCE:UNIPROT/SWISSPROT;ACC:O15496] Description

    Gene Info:
    Human Readable Name DRUGGABLE GENOME

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: January-2014

    Alternate Names:
    PLA2G10 Gene Symbol

    Gene Info:
    Target Class Enzymes
    Target Subclass EC:3.1.1.4

    Publications:

    • Version: 11-September-2012

    Alternate Names:
    PLA2G10 Uniprot Gene Name
    O15496 Uniprot Accession
    PA2GX_HUMAN Uniprot Id

    Gene Info:
    Uniprot Status Swiss-Prot
    Interpro Short Name PLipase_A2_euk
    Interpro Type Family

    Gene Categories:
    PHOSPHOLIPASE, DRUGGABLE GENOME

    Publications:

    • Version: chembl_23

    Alternate Names:
    PLA2G10 GENE_SYMBOL
    Group 10 secretory phospholipase A2 UNIPROT
    Group X secretory phospholipase A2 UNIPROT

    Gene Info:

    Publications:

    • Version: 31-May-2017

    Alternate Names:
    ENSG00000069764 Gene Symbol
    PLA2G10 Ensembl Id

    Gene Info:

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: 01-February-2022

    Alternate Names:
    Group 10 secretory phospholipase A2 Gene Name
    O15496 UniProt ID

    Gene Info:

    Gene Categories:
    ENZYME

    Publications:

    • Version: 01-February-2022

    Alternate Names:

    Gene Info:

    Gene Categories:
    PHOSPHOLIPASE

    Publications: