5739 |
PROSTAGLANDIN I2 RECEPTOR |
PTGIR |
IP |
PRIPR |
600022 |
9602 |
ENSG00000160013 |
OTTHUMG00000183429 |
PGI2 receptor |
PGI receptor |
Prostacyclin receptor |
Prostanoid IP receptor |
P43119 |
PI2R_HUMAN |
PROSTACYCLIN RECEPTOR (PROSTANOID IP RECEPTOR) (PGI RECEPTOR) (PROSTAGLANDIN I2 RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P43119] |
PA291 |
T99954 |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000276 |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Name | GPCR, rhodopsin-like, 7TM |
Interpro Short Name | 7TM_GPCR_Rhodpsn |
Interpro Type | Family |
Uniprot Status | Swiss-Prot |
Human Readable Name | DRUGGABLE GENOME |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Target Subclass | GPCR |
Transmembrane Helix Count | 7 |
Target Class | Receptors |
Gene Biotype | PROTEIN_CODING |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
agonist (activating) |
Trial Name | selexipag, ACT-293987 |
Novel drug target | Established target |
Trial Name | NS-304 |
agonist (activating) |
Mechanism of Interaction | Prostanoid IP receptor agonist |
Direct Interaction | yes |
Trial Name | iloprost,Ventavis |
agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Prostanoid IP receptor agonist |
agonist (activating) |
Mechanism of Interaction | Prostanoid IP receptor agonist |
Direct Interaction | yes |
agonist (activating) |
Novel drug target | Established target |
Trial Name | beraprost |
agonist (activating) |
Mechanism of Interaction | Prostanoid IP receptor agonist |
Direct Interaction | yes |
n/a |
Trial Name | APL-202,Isprelor |
Novel drug target | Established target |
agonist (activating) |
Direct Interaction | yes |
Mechanism of Interaction | Prostanoid IP receptor agonist |
PTGIR | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
PROSTACYCLIN RECEPTOR (PROSTANOID IP RECEPTOR) (PGI RECEPTOR) (PROSTAGLANDIN I2 RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P43119] | Description |
ENSG00000160013 | Ensembl Gene Id |
PTGIR | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PTGIR | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Rhodopsin |
ENSG00000160013 | Ensembl Gene Id |
PI2R_HUMAN | Uniprot Id |
PTGIR | Uniprot Gene Name |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000276 |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
ENSG00000160013 | Ensembl Gene Id |
P43119 | Uniprot Accession |
PI2R_HUMAN | Uniprot Id |
Target Subclass | Rhodopsin |
Target Main Class | Receptors |
Target Subclass | GPCR |
PA291 | PharmGKB ID |
PTGIR | TTD Gene Abbreviation |
T99954 | TTD Target ID |
ENSG00000160013 | Gene Symbol |
PTGIR | Ensembl Id |
DRUGGABLE GENOME |
PRIPR | GENE_SYMBOL |
PTGIR | GENE_SYMBOL |
Prostacyclin receptor | UNIPROT |
5739 | Gene ID |
IP | dGene Synonym |
PRIPR | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |