5745 |
PARATHYROID HORMONE 1 RECEPTOR |
PTH1R |
PFE |
PTHR |
PTHR1 |
168468 |
9608 |
ENSG00000160801 |
OTTHUMG00000133515 |
PTH/PTHr receptor |
PTH/PTHrP type I receptor |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
PTH1 receptor |
Q03431 |
PARATHYROID HORMONE/PARATHYROID HORMONE-RELATED PEPTIDE RECEPTOR PRECURSOR (PTH/PTHR RECEPTOR) (PTH/PTHRP TYPE I RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:Q03431] |
PTH1R_HUMAN |
T67710 |
EKNS |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Secretin |
Human Readable Name | DRUGGABLE GENOME |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Name | GPCR, family 2, secretin-like |
Interpro Short Name | GPCR_2_secretin-like |
Interpro Acc | IPR000832 |
Interpro Type | Family |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Target Main Class | Receptors |
Transmembrane Helix Count | 7 |
Gene Biotype | PROTEIN_CODING |
G PROTEIN COUPLED RECEPTOR |
DRUGGABLE GENOME |
agonist (activating) |
binder |
Trial Name | teriparatide, inhaled AIR |
Novel drug target | Established target |
Trial Name | teriparatide, PTH1-34 nasal spray |
agonist (activating) |
Mechanism of Interaction | Parathyroid hormone receptor agonist |
Direct Interaction | yes |
agonist (activating) |
Mechanism of Interaction | Parathyroid hormone receptor agonist |
Direct Interaction | yes |
Trial Name | PREOS |
PTH1R | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
PTH1R | Gene Symbol |
PTHR1 | Gene Symbol |
Target Class | Receptors |
Target Subclass | GPCR |
Target Subclass | Secretin |
Q03431 | Uniprot Accession |
PTHR1 | Gene Symbol |
ENSG00000160801 | Ensembl Gene Id |
Target Subclass | Secretin |
Target Subclass | GPCR |
Target Main Class | Receptors |
PTHR1 | Display Id |
PARATHYROID HORMONE/PARATHYROID HORMONE-RELATED PEPTIDE RECEPTOR PRECURSOR (PTH/PTHR RECEPTOR) (PTH/PTHRP TYPE I RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:Q03431] | Description |
ENSG00000160801 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
PARATHYROID HORMONE/PARATHYROID HORMONE-RELATED PEPTIDE RECEPTOR | Uniprot Protein Name |
Q03431 | Uniprot Accession |
5745 | Entrez Gene Id |
Human Readable Name | G PROTEIN COUPLED RECEPTOR |
Interpro Name | GPCR, family 2, secretin-like |
Interpro Short Name | GPCR_2_secretin-like |
G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME |
ENSG00000160801 | Gene Symbol |
PTH1R | Ensembl Id |
DRUGGABLE GENOME |
PTHR1 | GENE_SYMBOL |
PTH1R | GENE_SYMBOL |
Parathyroid hormone/parathyroid hormone-related peptide receptor | UNIPROT |
5745 | Gene ID |
PFE | dGene Synonym |
PTHR | dGene Synonym |
G PROTEIN COUPLED RECEPTOR |
PTH1R | TTD Gene Abbreviation |
T67710 | TTD Target ID |