6256 |
RETINOID X RECEPTOR ALPHA |
RXRA |
NR2B1 |
180245 |
10477 |
ENSG00000186350 |
OTTHUMG00000020887 |
P19793 |
RXRA_HUMAN |
RETINOIC ACID RECEPTOR RXR-ALPHA (RETINOID X RECEPTOR ALPHA). [SOURCE:UNIPROT/SWISSPROT;ACC:P19793] |
RETINOIC ACID RECEPTOR RXR-ALPHA |
Nuclear receptor subfamily 2 group B member 1 |
PA34890 |
T13726 |
RXR-alpha |
RXRalpha |
Human Readable Name | DRUGGABLE GENOME |
Target Class | Receptors |
Target Subclass | Nuclear receptor |
Interpro Short Name | Nucl_hrmn_rcpt_lig-bd_core |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000536 |
Interpro Type | Domain |
Human Readable Name | NUCLEAR HORMONE RECEPTOR |
Interpro Name | Nuclear hormone receptor, ligand-binding, core |
Uniprot Status | Swiss-Prot |
Initial Gene Query | NR2B1 |
Counted Citations from 1950-2000 | 1276 |
Target Main Class | Receptors |
Gene Biotype | PROTEIN_CODING |
TRANSCRIPTION FACTOR COMPLEX |
NUCLEAR HORMONE RECEPTOR |
DRUGGABLE GENOME |
TRANSCRIPTION FACTOR |
activator (activating) |
agonist (activating) |
Novel drug target | Established target |
Trial Name | bexarotene,Targretin |
Notes |
agonist (activating) |
Mechanism of Interaction | Retinoid receptor agonist |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Retinoid X receptor alpha modulator |
Direct Interaction | yes |
agonist (activating) |
Mechanism of Interaction | Retinoid X receptor agonist |
Direct Interaction | yes |
agonist (activating) |
Mechanism of Interaction | Retinoid receptor agonist |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Retinoid receptor modulator |
Direct Interaction | yes |
RXRA | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
6256 | Entrez Gene ID |
Initial Gene Query | NR2B1 |
Counted Citations from 1950-2000 | 1276 |
NUCLEAR HORMONE RECEPTOR |
ENSG00000186350 | Ensembl Gene Id |
RETINOIC ACID RECEPTOR RXR-ALPHA | Uniprot Protein Name |
6256 | Entrez Gene Id |
Interpro Short Name | Nucl_hrmn_rcpt_lig-bd_core |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Acc | IPR000536 |
NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME |
RXRA | Display Id |
ENSG00000186350 | Ensembl Gene Id |
RETINOIC ACID RECEPTOR RXR-ALPHA (RETINOID X RECEPTOR ALPHA). [SOURCE:UNIPROT/SWISSPROT;ACC:P19793] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
RXRA | Gene Symbol |
Target Class | Receptors |
Target Subclass | Nuclear receptor |
RXRA_HUMAN | Uniprot Id |
6256 | Entrez Gene Id |
ENSG00000186350 | Ensembl Gene Id |
Target Main Class | Receptors |
Target Subclass | Nuclear receptor |
PA34890 | PharmGKB ID |
RXRA | Gene Symbol |
NR2B1 | GENE_SYMBOL |
RXRA | GENE_SYMBOL |
Retinoic acid receptor RXR-alpha | UNIPROT |
ENSG00000186350 | Gene Symbol |
RXRA | Ensembl Id |
DRUGGABLE GENOME |
NR2B1 | GO Gene Synonym |
TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR |
RXRA | Gene Symbol |
CLINICALLY ACTIONABLE |
6256 | Gene ID |
NR2B1 | dGene Synonym |
NUCLEAR HORMONE RECEPTOR |
RXRA | TTD Gene Abbreviation |
T13726 | TTD Target ID |
Retinoic acid receptor RXR-alpha | Gene Name |
P19793 | UniProt ID |
NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR |