6559 |
SOLUTE CARRIER FAMILY 12 MEMBER 3 |
SLC12A3 |
NCC |
NCCT |
TSC |
600968 |
10912 |
ENSG00000070915 |
OTTHUMG00000133284 |
P55017 |
NA-CL SYMPORTER |
THIAZIDE-SENSITIVE SODIUM-CHLORIDE COTRANSPORTER |
S12A3_HUMAN |
Na-Cl cotransporter |
PA321 |
SOLUTE CARRIER FAMILY 12, MEMBER 3 (THIAZIDE-SENSITIVE SODIUM-CHLORIDE COTRANSPORTER) (NA-CL SYMPORTER). [SOURCE:UNIPROT/SWISSPROT;ACC:P55017] |
T84886 |
Target Class | Transporters |
Target Subclass | TC:2.A.30.4.2 |
Interpro Name | Thiazide-sensitive Na-K-Cl co-transporter |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Status | Swiss-Prot |
Interpro Short Name | NaCl_cotranspt |
Interpro Acc | IPR002948 |
Interpro Type | Domain |
Interpro Name | Amino acid permease domain |
Human Readable Name | TRANSPORTER |
Interpro Acc | IPR004841 |
Interpro Short Name | AA-permease_dom |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Type | Family |
Target Main Class | Transporters |
Target Subclass | SLC |
Transmembrane Helix Count | 12 |
Target Subclass | APC |
Target Subclass | SLC12 |
Gene Biotype | PROTEIN_CODING |
TRANSPORTER |
DRUGGABLE GENOME |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
Trial Name | - |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
Novel drug target | Established target |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
Trial Name | - |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
n/a |
Novel drug target | Established target |
Trial Name | - |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
Trial Name | Amturnide |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Thiazide-sensitive sodium-chloride cotransporter inhibitor |
Direct Interaction | yes |
SLC12A3 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
SOLUTE CARRIER FAMILY 12, MEMBER 3 (THIAZIDE-SENSITIVE SODIUM-CHLORIDE COTRANSPORTER) (NA-CL SYMPORTER). [SOURCE:UNIPROT/SWISSPROT;ACC:P55017] | Description |
ENSG00000070915 | Ensembl Gene Id |
SLC12A3 | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
SLC12A3 | Gene Symbol |
Target Class | Transporters |
Target Subclass | TC:2.A.30.4.2 |
S12A3_HUMAN | Uniprot Id |
P55017 | Uniprot Accession |
SLC12A3 | Gene Symbol |
Target Main Class | Transporters |
Target Subclass | SLC |
Transmembrane Helix Count | 12 |
P55017 | Uniprot Accession |
S12A3_HUMAN | Uniprot Id |
6559 | Entrez Gene Id |
Interpro Name | Thiazide-sensitive Na-K-Cl co-transporter |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Status | Swiss-Prot |
TRANSPORTER, DRUGGABLE GENOME |
PA321 | PharmGKB ID |
ENSG00000070915 | Gene Symbol |
SLC12A3 | Ensembl Id |
DRUGGABLE GENOME |
TSC | GENE_SYMBOL |
SLC12A3 | GENE_SYMBOL |
Solute carrier family 12 member 3 | UNIPROT |
SLC12A3 | TTD Gene Abbreviation |
T84886 | TTD Target ID |