706 |
TRANSLOCATOR PROTEIN |
TSPO |
BPBS |
BZRP |
DBI |
IBP |
MBR |
PBR |
PBS |
PKBS |
PTBR |
mDRC |
pk18 |
109610 |
1158 |
ENSG00000100300 |
OTTHUMG00000150573 |
P30536 |
PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR (PBR) (PKBS) (MITOCHONDRIAL BENZODIAZEPINE RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P30536] |
TSPOA_HUMAN |
T75440 |
Human Readable Name | DRUGGABLE GENOME |
Transmembrane Helix Count | 5 |
Target Subclass | Other |
Target Main Class | Transporters |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | TspO_MBR |
Interpro Name | TspO/MBR-related protein |
Interpro Type | Family |
Interpro Acc | IPR004307 |
Target Class | Transporters |
Target Subclass | Miscellaneous |
Target Subclass | benzodiazepine translocator protein, |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
n/a |
Trial Name | TLN-4601, ECO-4601 |
Novel drug target | Established target |
agonist (activating) |
Trial Name | - |
Novel drug target | Established target |
n/a |
Trial Name | AZ-007, Staccato zaleplon |
Novel drug target | Established target |
Trial Name | SKP-1041, delayed-release zaleplon |
n/a |
Trial Name | olesoxime, TRO19622 |
Novel drug target | Established target |
agonist (activating) |
Trial Name | - |
Novel drug target | Established target |
TSPO | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
TSPOA_HUMAN | Uniprot Id |
706 | Entrez Gene Id |
BZRP | Gene Symbol |
Transmembrane Helix Count | 5 |
Target Subclass | Other |
Target Main Class | Transporters |
TSPO | Gene Symbol |
BZRP | Gene Symbol |
Target Class | Transporters |
Target Subclass | Miscellaneous |
Target Subclass | benzodiazepine translocator protein, |
PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR (PBR) (PKBS) (MITOCHONDRIAL BENZODIAZEPINE RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:P30536] | Description |
BZRP | Display Id |
ENSG00000100300 | Ensembl Gene Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
TRANSLOCATOR PROTEIN | Uniprot Protein Name |
706 | Entrez Gene Id |
TSPO | Uniprot Gene Name |
Uniprot Status | Swiss-Prot |
Uniprot Evidence | 1: Evidence at protein level |
Interpro Short Name | TspO_MBR |
DRUGGABLE GENOME |
ENSG00000100300 | Gene Symbol |
TSPO | Ensembl Id |
DRUGGABLE GENOME |
TSPO | TTD Gene Abbreviation |
T75440 | TTD Target ID |