7422 |
VASCULAR ENDOTHELIAL GROWTH FACTOR A |
VEGFA |
MVCD1 |
VEGF |
VPF |
192240 |
12680 |
ENSG00000112715 |
OTTHUMG00000014745 |
P15692 |
VEGF-A |
Vascular permeability factor |
VEGFA_HUMAN |
PA37302 |
VASCULAR ENDOTHELIAL GROWTH FACTOR |
T96721 |
T20761 |
6071 |
Target Subclass | Growth factor |
Target Class | Ligand |
Target Subclass | Ligand |
Target Main Class | Other |
Gene Biotype | PROTEIN_CODING |
CELL SURFACE |
GROWTH FACTOR |
DRUGGABLE GENOME |
CLINICALLY ACTIONABLE |
inhibitor (inhibitory) |
Mechanism of Interaction | Vascular endothelial growth factor A inhibitor |
Direct Interaction | yes |
Trial Name | Lucentis |
n/a |
Trial Name | bevasiranib, Cand5 |
Novel drug target | Established target |
antagonist (inhibitory) |
Trial Name | Macugen |
Novel drug target | Established target |
Mechanism of Interaction | Vascular endothelial growth factor A antagonist |
antibody (inhibitory) |
binder |
inhibitor (inhibitory) |
Mechanism of Interaction | Vascular endothelial growth factor A inhibitor |
Direct Interaction | yes |
Trial Name | AVE-0005 |
inhibitor (inhibitory) |
Mechanism of Interaction | Vascular endothelial growth factor A inhibitor |
Direct Interaction | yes |
n/a |
Mechanism of Interaction | Vascular endothelial growth factor A binding agent |
Direct Interaction | yes |
antibody (inhibitory) |
inhibitor (inhibitory) |
Trial Name | Avastin |
Novel drug target | Established target |
Notes |
antibody (inhibitory) |
Notes | Fusion protein of extracellular domain portions from VEGFR-1 and VEGFR-2 combined with FC of human IGG |
inhibitor (inhibitory) |
Mechanism of Interaction | Vascular endothelial growth factor A inhibitor |
Direct Interaction | yes |
n/a |
Trial Name | 4SC-203 |
Novel drug target | Established target |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Vascular endothelial growth factor A inhibitor |
n/a |
VEGFA | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
VEGFA | Gene Symbol |
Target Class | Ligand |
Target Subclass | Ligand |
Target Subclass | Growth factor |
P15692 | Uniprot Accession |
VEGFA_HUMAN | Uniprot Id |
VEGF | Gene Symbol |
Target Subclass | Ligand |
Target Subclass | Growth factor |
Target Main Class | Other |
PA37302 | PharmGKB ID |
7422 | Entrez Gene ID |
6071 | CIViC Gene ID |
VEGFA | TTD Gene Abbreviation |
T20761 | TTD Target ID |
7422 | Entrez Gene Id |
VEGFA | MyCancerGenome Gene Symbol |
VEGFA | MyCancerGenome Reported Gene Name |
VEGF-A | Gene Symbol |
ENSG00000112715 | Gene Symbol |
VEGFA | Ensembl Id |
DRUGGABLE GENOME |
VEGF-A | UNIPROT |
VEGF | GENE_SYMBOL |
VEGFA | GENE_SYMBOL |
VEGF | Gene Symbol |
VEGF | GO Gene Synonym |
CELL SURFACE, GROWTH FACTOR |
VEGFA | Gene Symbol |
CLINICALLY ACTIONABLE |
VEGF | TTD Gene Abbreviation |
T96721 | TTD Target ID |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |