79001 |
VITAMIN K EPOXIDE REDUCTASE COMPLEX SUBUNIT 1 |
VKORC1 |
EDTP308 |
MST134 |
MST576 |
VKCFD2 |
VKOR |
608547 |
23663 |
ENSG00000167397 |
OTTHUMG00000047408 |
Q9BQB6 |
VITAMIN K1 2,3-EPOXIDE REDUCTASE SUBUNIT 1 |
UNQ308/PRO351 |
MSTP576 |
VKOR1_HUMAN |
PA133787052 |
Vitamin K epoxide reductase complex 1 |
T11843 |
Target Class | Enzymes |
Target Subclass | EC:1.1.4.1 |
Transmembrane Helix Count | 5 |
Target Main Class | Enzymes |
Target Subclass | 1.1 |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
ENZYME |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
inhibitor (inhibitory) |
Trial Name | - |
Novel drug target | Established target |
Mechanism of Interaction | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor |
n/a |
Trial Name | tecarfarin, ATI-5923 |
Novel drug target | Established target |
inhibitor (inhibitory) |
Mechanism of Interaction | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor |
Direct Interaction | yes |
Trial Name | - |
inhibitor (inhibitory) |
Mechanism of Interaction | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor |
VKORC1 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
VKORC1 | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:1.1.4.1 |
Q9BQB6 | Uniprot Accession |
ENSG00000167397 | Ensembl Gene Id |
79001 | Entrez Gene Id |
Transmembrane Helix Count | 5 |
Target Main Class | Enzymes |
Target Subclass | 1.1 |
PA133787052 | PharmGKB ID |
VKOR | GENE_SYMBOL |
MSTP576 | GENE_SYMBOL |
UNQ308/PRO351 | GENE_SYMBOL |
ENSG00000167397 | Gene Symbol |
VKORC1 | Ensembl Id |
DRUGGABLE GENOME |
VKORC1 | TTD Gene Abbreviation |
T11843 | TTD Target ID |
Vitamin K epoxide reductase complex subunit 1 | Gene Name |
Q9BQB6 | UniProt ID |
ENZYME |