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BUPRANOLOL Drug Record

  • Summary
  • Interactions
  • Claims
  • BUPRANOLOL chembl:CHEMBL305380

    Alternate Names:

    B-1312 [AS HYDROCHLORIDE]
    BUPRANOLOL HCL
    BUPRANOL
    KL-255 [AS HYDROCHLORIDE]
    BUPRANOLOL

    Drug Info:

    (0 More Sources)

    Publications:

    el Tayar N et al., 1988, Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists., J Med Chem
    Lenard et al., 2003, Activation of beta2- and beta3-adrenergic receptors increases brain tryptophan., J. Pharmacol. Exp. Ther.
    Zelaszczyk et al., 2009, Four close bupranolol analogues are antagonists at the low-affinity state of beta1-adrenoceptors., J. Physiol. Pharmacol.
  • BUPRANOLOL   ADRB1

    Interaction Score: 1.12

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:

    PMIDs:
    2903243 19439807


    Sources:
    DTC

  • BUPRANOLOL   ADRB2

    Interaction Score: 0.72

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:

    PMIDs:
    2903243 12606631


    Sources:
    DTC

  • DTC: BUPRANOLOL

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL305380 ChEMBL Drug ID

    Drug Info:

    Publications:
    el Tayar N et al., 1988, Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists., J Med Chem

  • ChemblDrugs: chembl:CHEMBL305380

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

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A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21