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CHEMBL261454 Drug Record

  • Summary
  • Interactions
  • Claims
  • CHEMBL261454 chembl:CHEMBL261454

    Alternate Names:

    HTS-466284
    LY-364947

    Drug Info:

    (0 More Sources)

    Publications:

    Bamborough et al., 2008, Assessment of chemical coverage of kinome space and its implications for kinase drug discovery., J. Med. Chem.
    Berman et al., 2000, The Protein Data Bank., Nucleic Acids Res.
  • CHEMBL261454   GAK

    Interaction Score: 15.46

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:

    PMIDs:
    19035792


    Sources:
    DTC

  • CHEMBL261454   CSNK1E

    Interaction Score: 10.3

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:

    PMIDs:
    19035792


    Sources:
    DTC

  • CHEMBL261454   TGFBR1

    Interaction Score: 7.73

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:

    PMIDs:
    19035792 10592235


    Sources:
    DTC

  • CHEMBL261454   CSNK1D

    Interaction Score: 1.47

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:

    PMIDs:
    19035792


    Sources:
    DTC

  • DTC: HTS-466284

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL261454 ChEMBL Drug ID

    Drug Info:

    Publications:
    Bamborough et al., 2008, Assessment of chemical coverage of kinome space and its implications for kinase drug discovery., J. Med. Chem.

  • ChemblDrugs: chembl:CHEMBL261454

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

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A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21