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DELAVIRDINE Drug Record

  • Summary
  • Interactions
  • Claims
  • DELAVIRDINE chembl:CHEMBL593 Approved

    Alternate Names:

    DELAVIRDINE
    U-90152
    N-{2-[4-(3-ISOPROPYLAMINO-PYRIDIN-2-YL)-PIPERAZINE-1-CARBONYL]-1H-INDOL-5-YL}-METHANESULFONAMIDE
    1-(3-((1-METHYLETHYL)AMINO)-2-PYRIDINYL)-4-((5-((METHYLSULFONYL)AMINO)-1H-INDOL-2-YL)CARBONYL)PIPERAZINE
    DELAVIRDINUM
    N-(2-(1-(3-(ISOPROPYLAMINO)PYRIDIN-2-YL)PIPERAZINE-4-CARBONYL)-1H-INDOL-5-YL)METHANESULFONAMIDE
    RESCRIPTOR
    DELAVIRDIN
    (N-[2-[4-[3-(1-METHYLETHYLAMINO)PYRIDIN-2-YL]PIPERAZIN-1-YL]CARBONYL-1H-INDOL-5-YL] METHANESULFONAMIDE)
    2-(4-(5-METHANESULFONAMIDO-1H-INDOL-2-YLCARBONYL)-1-PIPERAZINYL)-N-(1-METHYLETHYL)-3-PYRIDINAMINE
    DELAVIRDINA
    drugbank:00705
    chemidplus:136817-59-9
    rxcui:83816
    pubchem.compound:5625
    chembl:CHEMBL593

    Drug Info:

    (0 More Sources)

    Publications:

    Zembruski NC et al., 2011, Interaction potential of etravirine with drug transporters assessed in vitro., Antimicrob Agents Chemother
    Weiss J et al., 2007, Inhibition of MRP1/ABCC1, MRP2/ABCC2, and MRP3/ABCC3 by nucleoside, nucleotide, and non-nucleoside reverse transcriptase inhibitors., Drug Metab Dispos
  • DELAVIRDINE   ABCC3

    Interaction Score: 0.99

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    17172311


    Sources:
    DTC

  • DELAVIRDINE   ABCC1

    Interaction Score: 0.49

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    17172311


    Sources:
    DTC

  • DELAVIRDINE   ABCC2

    Interaction Score: 0.47

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    17172311


    Sources:
    DTC

  • DELAVIRDINE   ABCG2

    Interaction Score: 0.4

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    21189339


    Sources:
    DTC

  • DELAVIRDINE   ABCB1

    Interaction Score: 0.1

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    21189339


    Sources:
    DTC

  • DTC: DELAVIRDINE

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL593 ChEMBL Drug ID

    Drug Info:

    Publications:
    Weiss J et al., 2007, Inhibition of MRP1/ABCC1, MRP2/ABCC2, and MRP3/ABCC3 by nucleoside, nucleotide, and non-nucleoside reverse transcriptase inhibitors., Drug Metab Dispos
    Zembruski NC et al., 2011, Interaction potential of etravirine with drug transporters assessed in vitro., Antimicrob Agents Chemother

  • TTD: Delavirdine

    • Version: 2020.06.01

    Alternate Names:
    D0G6SD TTD Drug ID

    Drug Info:

    Publications:

  • ChemblDrugs: chembl:CHEMBL593

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

Disclaimer: This resource is intended for purely research purposes. It should not be used for emergencies or medical or professional advice.

A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21