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METRIBOLONE Drug Record

  • Summary
  • Interactions
  • Claims
  • METRIBOLONE chembl:CHEMBL166444

    Alternate Names:

    METHYLTRIENOLONE
    METRIBOLONE
    R-1881

    Drug Info:

    Drug Categories fused-ring compounds
    (0 More Sources)

    Publications:

    Berman et al., 2000, The Protein Data Bank., Nucleic Acids Res.
    Overington et al., 2006, How many drug targets are there?, Nat Rev Drug Discov
    Imming et al., 2006, Drugs, their targets and the nature and number of drug targets., Nat Rev Drug Discov
    Takeda AN et al., 2007, The synthetic androgen methyltrienolone (r1881) acts as a potent antagonist of the mineralocorticoid receptor., Mol Pharmacol
  • METRIBOLONE   NCOA2

    Interaction Score: 1.67

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    10592235


    Sources:
    DrugBank

  • METRIBOLONE   NR3C2

    Interaction Score: 0.98

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    17105867


    Sources:
    DrugBank

  • METRIBOLONE   PGR

    Interaction Score: 0.79

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    10592235 17139284 17016423


    Sources:
    DrugBank

  • METRIBOLONE   AR

    Interaction Score: 0.05

    Interaction Types & Directionality:
    agonist (activating)

    Interaction Info:
    Direct Interaction? False
    Specific Action of the Ligand Agonist
    Endogenous Drug? False

    PMIDs:
    10592235


    Sources:
    DrugBank GuideToPharmacology

  • DrugBank: DB02998

    • Version: 5.1.7

    Alternate Names:
    METRIBOLONE DrugBank Drug Name
    965-93-5 CAS Number
    CHEMBL166444 ChEMBL ID

    Drug Info:
    Drug Type small molecule
    Drug Groups experimental
    Drug Categories estranes

    Publications:
    Berman et al., 2000, The Protein Data Bank., Nucleic Acids Res.
    Takeda AN et al., 2007, The synthetic androgen methyltrienolone (r1881) acts as a potent antagonist of the mineralocorticoid receptor., Mol Pharmacol
    Overington et al., 2006, How many drug targets are there?, Nat Rev Drug Discov

  • GuideToPharmacology: 135650595

    • Version: 29-September-2020

    Alternate Names:
    METHYLTRIENOLONE GuideToPharmacology Ligand Name

    Drug Info:

    Publications:

  • ChemblDrugs: chembl:CHEMBL166444

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

Disclaimer: This resource is intended for purely research purposes. It should not be used for emergencies or medical or professional advice.

A finding of a drug-gene interaction or potentially druggable category does not necessarily indicate effectiveness (or lack thereof) of any drug or treatment regimen. A finding of no interaction or no potentially druggable category does not necessarily indicate lack of effectiveness of any drug or treatment regimen. Drug-gene interactions or potentially druggable categories are not presented in ranked order of potential or predicted efficacy.

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DGIdb (v4.2.0 - sha1 afd9f30b) • Last updated 2020-10-21