• Interaction Score: 0.46

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Details of the Assay for Interaction Determined from a radioligand binding assay using membranes from CHO‐K1 cells expressing the hM<sub>1</sub> receptor, and displacement of [<sup>3</sup>H]NMS tracer.
    Specific Action of the Ligand Antagonist
    Endogenous Drug? False

  • Interaction Score: 0.22

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Details of the Assay for Interaction Determined from a radioligand binding assay using membranes from CHO‐K1 cells expressing the hM<sub>4</sub> receptor, and displacement of [<sup>3</sup>H]NMS tracer.
    Specific Action of the Ligand Antagonist
    Endogenous Drug? False

    PMIDs:
    None found


  • Interaction Score: 0.2

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Details of the Assay for Interaction Determined from a radioligand binding assay using membranes from CHO‐K1 cells expressing the hM<sub>5</sub> receptor, and displacement of [<sup>3</sup>H]NMS tracer.
    Specific Action of the Ligand Antagonist
    Endogenous Drug? False

    PMIDs:
    None found


  • Interaction Score: 0.15

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Details of the Assay for Interaction Determined from a radioligand binding assay using membranes from CHO‐K1 cells expressing the hM<sub>2</sub> receptor, and displacement of [<sup>3</sup>H]NMS tracer.
    Specific Action of the Ligand Antagonist
    Endogenous Drug? False

    PMIDs:
    None found


  • Interaction Score: 0.13

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Details of the Assay for Interaction Determined from a radioligand binding assay using membranes from CHO‐K1 cells expressing the hM<sub>3</sub> receptor, and displacement of [<sup>3</sup>H]NMS tracer.
    Specific Action of the Ligand Antagonist
    Endogenous Drug? False

    PMIDs:
    None found


    • Version: 2020.06.01

    Alternate Names:
    D0XV4Z TTD Drug ID

    Drug Info:

    Publications:

    • Version: 2020.06.01

    Alternate Names:
    D0K1ST TTD Drug ID

    Drug Info:

    Publications:

    • Version: 29-September-2020

    Alternate Names:
    REVEFENACIN GuideToPharmacology Ligand Name

    Drug Info:

    Publications:

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications: