• Interaction Score: 1.82

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Trial Name AZ-007, Staccato zaleplon
    Novel drug target Established target
    Trial Name SKP-1041, delayed-release zaleplon

  • Interaction Score: 1.7

    Interaction Types & Directionality:
    positive modulator (activating)
    potentiator

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator
    Trial Name AZ-007, Staccato zaleplon

  • Interaction Score: 0.25

    Interaction Types & Directionality:
    positive modulator (activating)

    Interaction Info:
    Mechanism of Interaction GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.23

    Interaction Types & Directionality:
    positive modulator (activating)

    Interaction Info:
    Mechanism of Interaction GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator
    Direct Interaction yes

    PMIDs:
    None found


    • Version: 01-August-2011

    Alternate Names:
    ZALEPLON Primary Drug Name

    Drug Info:
    Year of Approval 1999
    Drug Class hypnotics and sedatives

    Publications:

    • Version: January-2014

    Alternate Names:

    Drug Info:
    Drug Indications hypnotic
    Drug Class Small Molecule
    FDA Approval approved

    Publications:

    • Version: 2020.06.01

    Alternate Names:
    D09DWL TTD Drug ID

    Drug Info:

    Publications:

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications:

    • Version: chembl_23

    Alternate Names:

    Drug Info:

    Publications: