23476 |
BROMODOMAIN CONTAINING 4 |
BRD4 |
CAP |
HUNK1 |
HUNKI |
MCAP |
608749 |
13575 |
ENSG00000141867 |
OTTHUMG00000183252 |
1945 |
NM_058243 |
NP_490597 |
O60885 |
9588 |
Bromodomain-containing protein 4 |
T40556 |
GuideToPharmacology Gene Category Name | Bromodomain kinase (BRDK) family |
GuideToPharmacology Gene Category ID | 558 |
Gene Biotype | PROTEIN_CODING |
KINASE |
SERINE THREONINE KINASE |
DRUGGABLE GENOME |
CLINICALLY ACTIONABLE |
ENZYME |
inhibitor (inhibitory) |
Details of the Assay for Interaction | Displacement of a tetra-acetylated histone H4 peptide from the tandem BET bromodomains of BRD4. |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
inhibitor (inhibitory) |
Direct Interaction? | False |
Endogenous Drug? | False |
Specific Action of the Ligand | Inhibition |
inhibitor (inhibitory) |
Details of the Assay for Interaction | Displacement of a tetra-acetylated histone H4 peptide from the tandem BET bromodomains of BRD4. |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
inhibitor (inhibitory) |
Direct Interaction? | False |
Endogenous Drug? | False |
Specific Action of the Ligand | Inhibition |
inhibitor (inhibitory) |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
Direct Interaction? | False |
inhibitor (inhibitory) |
Specific Action of the Ligand | Inhibition |
Endogenous Drug? | False |
Direct Interaction? | False |
BRD4 | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
13575 | HUGO Gene ID |
13575 | HUGO Gene Symbol |
bromodomain containing 4 | HUGO Gene Name |
GuideToPharmacology Gene Category Name | Bromodomain kinase (BRDK) family |
GuideToPharmacology Gene Category ID | 558 |
ENZYME |
23476 | Entrez Gene ID |
9588 | CIViC Gene ID |
ENSG00000141867 | Gene Symbol |
BRD4 | Ensembl Id |
DRUGGABLE GENOME |
Bromodomain-containing protein 4 | Gene Name |
O60885 | UniProt ID |
KINASE |
BRD4 | Gene Symbol |
CLINICALLY ACTIONABLE |
23476 | Gene ID |
CAP | dGene Synonym |
HUNK1 | dGene Synonym |
KINASE, SERINE THREONINE KINASE |
BRD4 | TTD Gene Abbreviation |
T40556 | TTD Target ID |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |
CLINICALLY ACTIONABLE |