DGIdb - THIOPERAMIDE Drug Record

THIOPERAMIDE chembl:CHEMBL260374

Alternate Names:

THIOPERAMIDE

Drug Info:

(0 More Sources)

Publications:

Smits RA et al., 2010, Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists., J Med Chem
Smits RA et al., 2008, Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach., J Med Chem

THIOPERAMIDE HRH4

Interaction Score: 3.09

Interaction Types & Directionality:

antagonist (inhibitory)

Interaction Info:

PMIDs:
20192225 19053770

Sources:
DTC
THIOPERAMIDE CYP2C9

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
THIOPERAMIDE CYP2C19

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
THIOPERAMIDE CYP1A2

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
THIOPERAMIDE CYP2D6

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
THIOPERAMIDE CYP3A4

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

DTC: THIOPERAMIDE

Version: 02-September-2020

Alternate Names:

CHEMBL260374 ChEMBL Drug ID

Drug Info:

Publications:

Smits RA et al., 2008, Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach., J Med Chem

Smits RA et al., 2010, Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists., J Med Chem

ChemblDrugs: chembl:CHEMBL260374
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:

THIOPERAMIDE Drug Record

THIOPERAMIDE chembl:CHEMBL260374

Alternate Names:

Drug Info:

Publications:

THIOPERAMIDE HRH4

Interaction Types & Directionality: antagonist (inhibitory)

Interaction Info:

PMIDs: 20192225 19053770

Sources: DTC

THIOPERAMIDE CYP2C9

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

THIOPERAMIDE CYP2C19

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

THIOPERAMIDE CYP1A2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

THIOPERAMIDE CYP2D6

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

THIOPERAMIDE CYP3A4

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

DTC: THIOPERAMIDE

Alternate Names: CHEMBL260374 ChEMBL Drug ID

Drug Info:

Publications: Smits RA et al., 2008, Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach., J Med Chem Smits RA et al., 2010, Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists., J Med Chem

ChemblDrugs: chembl:CHEMBL260374

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

antagonist (inhibitory)

PMIDs:
20192225 19053770

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Alternate Names:

CHEMBL260374 ChEMBL Drug ID

Publications:

Smits RA et al., 2008, Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach., J Med Chem

Smits RA et al., 2010, Synthesis and QSAR of quinazoline sulfonamides as highly potent human histamine H4 receptor inverse agonists., J Med Chem