• VARLITINIB chembl:CHEMBL2103842 Antineoplastic

    Alternate Names:

    AR-00334543
    ARRY-334543
    VARLITINIB
    ARRY-543
    ASLAN-001
    ASLAN001

    Drug Info:

    FDA Approval not approved
    Drug Class Small molecule
    Drug Indications antineoplastic agent
    (1 More Sources)

    Publications:

  • Interaction Score: 0.84

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Novel drug target Established target
    Trial Name ARRY-334543
    combination therapy trastuzumab + varlitinib

    PMIDs:
    None found


  • Interaction Score: 0.55

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Trial Name ARRY-334543
    Novel drug target Established target
    Mechanism of Interaction Epidermal growth factor receptor erbB1 inhibitor

    PMIDs:
    None found