• MAP3K5 4217 Druggable Genome

    Alternate Names:

    4217
    MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 5
    MAP3K5
    ASK1
    MAPKKK5
    MEKK5
    602448
    6857
    ENSG00000197442
    OTTHUMG00000015647
    Q99683
    MAPK/ERK kinase kinase 5
    MEKK 5
    MEK kinase 5
    Apoptosis signal-regulating kinase 1
    ASK-1
    MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 5 (EC 2.7.1.37) (MAPK/ERK KINASE KINASE 5) (MEK KINASE 5) (MEKK 5) (APOPTOSIS SIGNAL- REGULATING KINASE 1) (ASK-1). [SOURCE:UNIPROT/SWISSPROT;ACC:Q99683]
    M3K5_HUMAN
    PA30601
    T97589

    Gene Info:

    Human Readable Name DRUGGABLE GENOME
    Interpro Type Domain
    Interpro Acc IPR002290
    Interpro Name Serine/threonine- / dual-specificity protein kinase, catalytic domain
    Interpro Short Name Ser/Thr_dual-sp_kinase_dom
    Human Readable Name KINASE
    Uniprot Status Swiss-Prot
    Uniprot Evidence 1: Evidence at protein level
    Gene Biotype PROTEIN_CODING
    (6 More Sources)

    Gene Categories: Category Details

    KINASE
    SERINE THREONINE KINASE
    EXTERNAL SIDE OF PLASMA MEMBRANE
    DRUGGABLE GENOME
    TRANSCRIPTION FACTOR
  • Interaction Score: 61.83

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Mitogen-activated protein kinase kinase kinase 5 inhibitor
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 4.42

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    23556445


    Sources:
    PharmGKB

    • Version: 101_38

    Alternate Names:
    MAP3K5 Ensembl Gene Name

    Gene Info:
    Gene Biotype PROTEIN_CODING

    Publications:

    • Version: 26-July-2011

    Alternate Names:
    MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 5 (EC 2.7.1.37) (MAPK/ERK KINASE KINASE 5) (MEK KINASE 5) (MEKK 5) (APOPTOSIS SIGNAL- REGULATING KINASE 1) (ASK-1). [SOURCE:UNIPROT/SWISSPROT;ACC:Q99683] Description
    MAP3K5 Display Id
    ENSG00000197442 Ensembl Gene Id

    Gene Info:
    Human Readable Name DRUGGABLE GENOME

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: 11-September-2012

    Alternate Names:
    MAP3K5 Uniprot Gene Name
    M3K5_HUMAN Uniprot Id
    Q99683 Uniprot Accession

    Gene Info:
    Interpro Type Domain
    Interpro Acc IPR002290
    Interpro Name Serine/threonine- / dual-specificity protein kinase, catalytic domain

    Gene Categories:
    KINASE, DRUGGABLE GENOME

    Publications:

    • Version: 18-August-2020
    • Version: 31-May-2017

    Alternate Names:
    ENSG00000197442 Gene Symbol
    MAP3K5 Ensembl Id

    Gene Info:

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: chembl_23

    Alternate Names:
    MEK kinase 5 UNIPROT
    MAPKKK5 GENE_SYMBOL
    MEKK5 GENE_SYMBOL

    Gene Info:

    Publications:

    • Version: 01-February-2022

    Alternate Names:
    ASK1 GO Gene Synonym
    MAPKKK5 GO Gene Synonym
    MEKK5 GO Gene Synonym

    Gene Info:

    Gene Categories:
    SERINE THREONINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE

    Publications:

    • Version: 27-Jun-2013

    Alternate Names:
    4217 Gene ID
    ASK1 dGene Synonym
    MAPKKK5 dGene Synonym

    Gene Info:

    Gene Categories:
    KINASE, SERINE THREONINE KINASE

    Publications:

  • Alternate Names:
    MAP3K5 TTD Gene Abbreviation
    T97589 TTD Target ID

    Gene Info:

    Publications:

    • Version: 01-February-2022

    Alternate Names:
    Mitogen-activated protein kinase kinase kinase 5 Gene Name
    Q99683 UniProt ID

    Gene Info:

    Gene Categories:
    KINASE, TRANSCRIPTION FACTOR

    Publications: