• PTGDR 5729 Druggable Genome

    Alternate Names:

    5729
    PROSTAGLANDIN D2 RECEPTOR
    PTGDR
    AS1
    ASRT1
    DP
    DP1
    PTGDR1
    604687
    9591
    ENSG00000168229
    OTTHUMG00000140299
    Q13258
    PROSTAGLANDIN D2 RECEPTOR (PROSTANOID DP RECEPTOR) (PGD RECEPTOR). [SOURCE:UNIPROT/SWISSPROT;ACC:Q13258]
    PGD2 receptor
    Prostanoid DP receptor
    PGD receptor
    PD2R_HUMAN
    PA285
    T68782

    Gene Info:

    Human Readable Name G PROTEIN COUPLED RECEPTOR
    Target Class Receptors
    Target Subclass GPCR
    Target Subclass Rhodopsin
    Human Readable Name DRUGGABLE GENOME
    Interpro Short Name 7TM_GPCR_Rhodpsn
    Uniprot Evidence 2: Evidence at transcript level
    Interpro Name GPCR, rhodopsin-like, 7TM
    Interpro Acc IPR000276
    Interpro Type Family
    Uniprot Status Swiss-Prot
    Gene Biotype PROTEIN_CODING
    (7 More Sources)

    Gene Categories: Category Details

    G PROTEIN COUPLED RECEPTOR
    DRUGGABLE GENOME
  • Interaction Score: 17.67

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Prostanoid DP receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 6.31

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Trial Name MK-0524A, ER niacin/laropiprant,Tredaptive, Trevaclyn, Pelzont
    Novel drug target Established target
    Trial Name MK-0542B, extended release niacin + laropiprant +simvastatin

  • Interaction Score: 4.42

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

  • Interaction Score: 4.42

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

  • Interaction Score: 4.42

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Prostanoid DP receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 4.42

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Novel drug target Established target
    Trial Name AM-461

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

  • Interaction Score: 4.42

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD