• Interaction Score: 46.37

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Novel drug target Novel Target
    Trial Name Saredutant, SR 48968

  • Interaction Score: 30.91

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Neurokinin 2 receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 15.46

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

  • Interaction Score: 3.86

    Interaction Types & Directionality:
    n/a

    Interaction Info:

    PMIDs:
    None found


    Sources:
    TTD

    • Version: 101_38

    Alternate Names:
    TACR2 Ensembl Gene Name

    Gene Info:
    Gene Biotype PROTEIN_CODING

    Publications:

    • Version: January-2014

    Alternate Names:
    TACR2 Gene Symbol

    Gene Info:
    Target Class Receptors
    Target Subclass GPCR
    Target Subclass Rhodopsin

    Publications:

    • Version: 11-September-2012

    Alternate Names:
    TACR2 Uniprot Gene Name
    P21452 Uniprot Accession
    6865 Entrez Gene Id

    Gene Info:
    Uniprot Status Swiss-Prot
    Interpro Type Family
    Uniprot Evidence 2: Evidence at transcript level

    Gene Categories:
    G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME

    Publications:

    • Version: 26-July-2011

    Alternate Names:
    TACR2 Display Id
    SUBSTANCE-K RECEPTOR (SKR) (NEUROKININ A RECEPTOR) (NK-2 RECEPTOR) (NK-2R) (TACHYKININ RECEPTOR 2). [SOURCE:UNIPROT/SWISSPROT;ACC:P21452] Description
    ENSG00000075073 Ensembl Gene Id

    Gene Info:
    Human Readable Name DRUGGABLE GENOME

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: 31-May-2017

    Alternate Names:
    ENSG00000075073 Gene Symbol
    TACR2 Ensembl Id

    Gene Info:

    Gene Categories:
    DRUGGABLE GENOME

    Publications:

    • Version: chembl_23

    Alternate Names:
    NKNAR GENE_SYMBOL
    TAC2R GENE_SYMBOL
    TACR2 GENE_SYMBOL

    Gene Info:

    Publications:

    • Version: 27-Jun-2013

    Alternate Names:
    6865 Gene ID
    NK2R dGene Synonym
    NKNAR dGene Synonym

    Gene Info:

    Gene Categories:
    G PROTEIN COUPLED RECEPTOR

    Publications:

    • Version: 2020.06.01

    Alternate Names:
    TACR2 TTD Gene Abbreviation
    T52790 TTD Target ID

    Gene Info:

    Publications: