DGIdb - CHEMBL59030 Drug Record

CHEMBL59030 chembl:CHEMBL59030

Alternate Names:

GW3965

Drug Info:

(0 More Sources)

Publications:

Chao EY et al., 2008, Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity., J Med Chem
Overington et al., 2006, How many drug targets are there?, Nat Rev Drug Discov
Imming et al., 2006, Drugs, their targets and the nature and number of drug targets., Nat Rev Drug Discov

CHEMBL59030 NR1H2

Interaction Score: 3.43

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
18800767 17139284 17016423

Sources:
DTC
CHEMBL59030 NR1H3

Interaction Score: 1.21

Interaction Types & Directionality:

agonist (activating)

Interaction Info:

PMIDs:
18800767

Sources:
DTC
CHEMBL59030 KAT2A

Interaction Score: 0.08

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
CHEMBL59030 RECQL

Interaction Score: 0.06

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
CHEMBL59030 VDR

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
CHEMBL59030 EHMT2

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

DTC: GW3965
- Version: 02-September-2020
Alternate Names:

CHEMBL59030 ChEMBL Drug ID

Drug Info:

Publications:

Chao EY et al., 2008, Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity., J Med Chem
ChemblDrugs: chembl:CHEMBL59030
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:

CHEMBL59030 Drug Record

CHEMBL59030 chembl:CHEMBL59030

Alternate Names:

Drug Info:

Publications:

CHEMBL59030 NR1H2

Interaction Types & Directionality: agonist (activating)

Interaction Info:

PMIDs: 18800767 17139284 17016423

Sources: DTC

CHEMBL59030 NR1H3

Interaction Types & Directionality: agonist (activating)

Interaction Info:

PMIDs: 18800767

Sources: DTC

CHEMBL59030 KAT2A

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

CHEMBL59030 RECQL

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

CHEMBL59030 VDR

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

CHEMBL59030 EHMT2

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

DTC: GW3965

Alternate Names: CHEMBL59030 ChEMBL Drug ID

Drug Info:

Publications: Chao EY et al., 2008, Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity., J Med Chem

ChemblDrugs: chembl:CHEMBL59030

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

agonist (activating)

PMIDs:
18800767 17139284 17016423

Sources:
DTC

Interaction Types & Directionality:

agonist (activating)

PMIDs:
18800767

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Alternate Names:

CHEMBL59030 ChEMBL Drug ID

Publications:

Chao EY et al., 2008, Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity., J Med Chem