• DEFACTINIB chembl:CHEMBL3137331 Antineoplastic

    Alternate Names:

    DEFACTINIB
    PF-04554878
    VS-6063

    Drug Info:

    FDA Approval not approved
    Drug Class small molecule
    Drug Indications antineoplastic agent
    (0 More Sources)

    Publications:

  • Interaction Score: 2.38

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Novel drug target Novel Target
    Trial Name PF-04554878
    Mechanism of Interaction Focal adhesion kinase 1 inhibitor

    PMIDs:
    None found


  • Interaction Score: 1.72

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Protein tyrosine kinase 2 beta inhibitor
    Direct Interaction yes

    PMIDs:
    None found