DGIdb - ESTRAMUSTINE Drug Record

ESTRAMUSTINE chembl:CHEMBL1575 AntineoplasticImmunotherapy

Alternate Names:

NSC-89201
RO-222296000
RO-22-2296000
ESTRAMUSTINE
ESTRACYT®
EMCYT®
ESTRADIOL 3-(N,N-BIS(2-CHLOROETHYL)CARBAMATE)
17Β-ESTRADIOL 3-(BIS(2-CHLOROETHYL)CARBAMATE)
17BETA-ESTRADIOL 3-(BIS(2-CHLOROETHYL)CARBAMATE)
ESTRAMUSTINUM
ESTRAMUSTINA
chemidplus:2998-57-4
drugbank:01196
chembl:CHEMBL1575
rxcui:4089
pubchem.compound:259331

Drug Info:

(0 More Sources)

Publications:

Peterson et al., 1981, Intracellular localization of estramustine in rat ventral prostate in vitro., Prostate
Serafin et al., Influence of p53 and bcl-2 on chemosensitivity in benign and malignant prostatic cell lines., Urol. Oncol.
Munshi et al., 2001, Chemotherapy in patients with prostate specific antigen-only disease after primary therapy for prostate carcinoma: a phase II trial of oral estramustine and oral etoposide., Cancer

ESTRAMUSTINE HEXB

Interaction Score: 1.25

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
6795611

Sources:
NCI
ESTRAMUSTINE KLK3

Interaction Score: 0.62

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
11391599

Sources:
NCI
ESTRAMUSTINE BCL2

Interaction Score: 0.26

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
15869997

Sources:
NCI
ESTRAMUSTINE BAX

Interaction Score: 0.23

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
15869997

Sources:
NCI
ESTRAMUSTINE TDP1

Interaction Score: 0.09

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE BLM

Interaction Score: 0.06

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE KAT2A

Interaction Score: 0.04

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE USP1

Interaction Score: 0.03

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE POLK

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE VDR

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
ESTRAMUSTINE AR

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

NCI: ESTRAMUSTINE

Version: 14-September-2017

Alternate Names:

C479 NCI drug code

Drug Info:

Publications:

Munshi et al., 2001, Chemotherapy in patients with prostate specific antigen-only disease after primary therapy for prostate carcinoma: a phase II trial of oral estramustine and oral etoposide., Cancer

Serafin et al., Influence of p53 and bcl-2 on chemosensitivity in benign and malignant prostatic cell lines., Urol. Oncol.

Peterson et al., 1981, Intracellular localization of estramustine in rat ventral prostate in vitro., Prostate

DTC: ESTRAMUSTINE
- Version: 02-September-2020
Alternate Names:

CHEMBL1575 ChEMBL Drug ID

Drug Info:

Publications:
TTD: Estramustine
- Version: 2020.06.01
Alternate Names:

D03SRY TTD Drug ID

Drug Info:

Publications:
ChemblDrugs: chembl:CHEMBL1575
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:

ESTRAMUSTINE Drug Record

ESTRAMUSTINE chembl:CHEMBL1575 AntineoplasticImmunotherapy

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 6795611

Sources: NCI

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 11391599

Sources: NCI

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 15869997

Sources: NCI

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 15869997

Sources: NCI

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

NCI: ESTRAMUSTINE

Alternate Names: C479 NCI drug code

Drug Info:

DTC: ESTRAMUSTINE

Alternate Names: CHEMBL1575 ChEMBL Drug ID

Drug Info:

Publications:

TTD: Estramustine

Alternate Names: D03SRY TTD Drug ID

Drug Info:

Publications:

ChemblDrugs: chembl:CHEMBL1575

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

n/a

PMIDs:
6795611

Sources:
NCI

Interaction Types & Directionality:

n/a

PMIDs:
11391599

Sources:
NCI

Interaction Types & Directionality:

n/a

PMIDs:
15869997

Sources:
NCI

Interaction Types & Directionality:

n/a

PMIDs:
15869997

Sources:
NCI

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Alternate Names:

C479 NCI drug code

Alternate Names:

CHEMBL1575 ChEMBL Drug ID

Alternate Names:

D03SRY TTD Drug ID