DGIdb - KETANSERIN Drug Record

KETANSERIN chembl:CHEMBL51 Approved

Alternate Names:

R-41468
KETANSERIN
SUFREXAL

Drug Info:

(0 More Sources)

Publications:

O'Neill et al., 1998, Effects of 5-hydroxytryptamine2 receptor antagonism on the behavioral activation and immediate early gene expression induced by dizocilpine., J. Pharmacol. Exp. Ther.
Lacivita E et al., 2012, Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo., J Med Chem
Kasho et al., 1998, Serotonin enhances the production of type IV collagen by human mesangial cells., Kidney Int.
Muntasir HA et al., 2006, Inverse agonist activity of sarpogrelate, a selective 5-HT2A-receptor antagonist, at the constitutively active human 5-HT2A receptor., J Pharmacol Sci

KETANSERIN HTR7

Interaction Score: 0.67

Interaction Types & Directionality:

antagonist (inhibitory)

Interaction Info:

PMIDs:
22738316

Sources:
DTC
KETANSERIN HSPA4

Interaction Score: 0.5

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
9864262

Sources:
NCI
KETANSERIN HTR2A

Interaction Score: 0.23

Interaction Types & Directionality:

inverse agonist (inhibitory)

antagonist (inhibitory)

Interaction Info:

PMIDs:
9767524 17031071

Sources:
NCI
KETANSERIN DRD1

Interaction Score: 0.05

Interaction Types & Directionality:

antagonist (inhibitory)

Interaction Info:

PMIDs:
None found

Sources:
DTC
KETANSERIN HPGD

Interaction Score: 0.03

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
KETANSERIN CYP2C9

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
KETANSERIN CYP2C19

Interaction Score: 0.02

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC
KETANSERIN EHMT2

Interaction Score: 0.01

Interaction Types & Directionality:

n/a

Interaction Info:

PMIDs:
None found

Sources:
DTC

NCI: KETANSERIN

Version: 14-September-2017

Alternate Names:

C604 NCI drug code

Drug Info:

Publications:

O'Neill et al., 1998, Effects of 5-hydroxytryptamine2 receptor antagonism on the behavioral activation and immediate early gene expression induced by dizocilpine., J. Pharmacol. Exp. Ther.

Kasho et al., 1998, Serotonin enhances the production of type IV collagen by human mesangial cells., Kidney Int.

DTC: KETANSERIN

Version: 02-September-2020

Alternate Names:

CHEMBL51 ChEMBL Drug ID

Drug Info:

Publications:

Lacivita E et al., 2012, Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo., J Med Chem

TTD: Ketanserin
- Version: 2020.06.01
Alternate Names:

D08VRO TTD Drug ID

Drug Info:

Publications:
ChemblDrugs: chembl:CHEMBL51
- Version: ChEMBL_27
Alternate Names:

Drug Info:

Publications:

inverse agonist (inhibitory)
antagonist (inhibitory)

KETANSERIN Drug Record

KETANSERIN chembl:CHEMBL51 Approved

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality: antagonist (inhibitory)

Interaction Info:

PMIDs: 22738316

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: 9864262

Sources: NCI

Interaction Types & Directionality: inverse agonist (inhibitory) antagonist (inhibitory)

Interaction Info:

PMIDs: 9767524 17031071

Sources: NCI

Interaction Types & Directionality: antagonist (inhibitory)

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

Interaction Types & Directionality: n/a

Interaction Info:

PMIDs: None found

Sources: DTC

NCI: KETANSERIN

Alternate Names: C604 NCI drug code

Drug Info:

DTC: KETANSERIN

Alternate Names: CHEMBL51 ChEMBL Drug ID

Drug Info:

Publications: Lacivita E et al., 2012, Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo., J Med Chem

TTD: Ketanserin

Alternate Names: D08VRO TTD Drug ID

Drug Info:

Publications:

ChemblDrugs: chembl:CHEMBL51

Alternate Names:

Drug Info:

Publications:

Interaction Types & Directionality:

antagonist (inhibitory)

PMIDs:
22738316

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
9864262

Sources:
NCI

Interaction Types & Directionality:

inverse agonist (inhibitory)

antagonist (inhibitory)

PMIDs:
9767524 17031071

Sources:
NCI

Interaction Types & Directionality:

antagonist (inhibitory)

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Interaction Types & Directionality:

n/a

PMIDs:
None found

Sources:
DTC

Alternate Names:

C604 NCI drug code

Alternate Names:

CHEMBL51 ChEMBL Drug ID

Publications:

Lacivita E et al., 2012, Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo., J Med Chem

Alternate Names:

D08VRO TTD Drug ID