• Interaction Score: 1.51

    Interaction Types & Directionality:
    agonist (activating)
    antagonist (inhibitory)

    Interaction Info:
    Trial Name nalmefene, CPH-101
    Novel drug target Established target

  • Interaction Score: 0.91

    Interaction Types & Directionality:
    partial agonist (activating)
    antagonist (inhibitory)

    Interaction Info:
    Trial Name nalmefene, CPH-101
    Novel drug target Established target

    PMIDs:
    9862779


  • Interaction Score: 0.2

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Novel drug target Established target
    Trial Name nalmefene, CPH-101

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

    • Version: January-2014

    Alternate Names:

    Drug Info:
    Drug Indications smoking-cessation agent,for treatment of addiction
    Drug Class Small molecule
    FDA Approval approved

    Publications:

    • Version: 02-September-2020

    Alternate Names:
    CHEMBL982 ChEMBL Drug ID

    Drug Info:

    Publications:

    • Version: 2020.06.01

    Alternate Names:
    D05VIL TTD Drug ID

    Drug Info:

    Publications:

    • Version: ChEMBL_27

    Alternate Names:

    Drug Info:

    Publications: