• TEDATIOXETINE chembl:CHEMBL2104986

    Alternate Names:

    TEDATIOXETINE
    LU-AA24530

    Drug Info:

    FDA Approval not approved
    Drug Class small molecule
    Drug Indications antidepressant
    (0 More Sources)

    Publications:

  • Interaction Score: 0.95

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Serotonin 3 (5-HT3) receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.95

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Serotonin 3 (5-HT3) receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.79

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction Serotonin 3 (5-HT3) receptor antagonist

    PMIDs:
    None found


  • Interaction Score: 0.4

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Mechanism of Interaction Serotonin 3 (5-HT3) receptor antagonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.32

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Novel drug target Established target
    Trial Name Lu AA24530
    Mechanism of Interaction Serotonin 3 (5-HT3) receptor antagonist

    PMIDs:
    None found


  • Interaction Score: 0.29

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Trial Name Lu AA24530
    Novel drug target Established target
    Mechanism of Interaction Serotonin 2c (5-HT2c) receptor antagonist

    PMIDs:
    None found


  • Interaction Score: 0.19

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Dopamine transporter inhibitor
    Direct Interaction yes
    Trial Name Lu AA24530

    PMIDs:
    None found


  • Interaction Score: 0.12

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Trial Name Lu AA24530
    Novel drug target Established target

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

  • Interaction Score: 0.11

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction Alpha-1a adrenergic receptor antagonist
    Trial Name Lu AA24530

    PMIDs:
    None found


  • Interaction Score: 0.09

    Interaction Types & Directionality:
    n/a

    Interaction Info:
    Trial Name Lu AA24530
    Novel drug target Established target

    PMIDs:
    None found


    Sources:
    TdgClinicalTrial

  • Interaction Score: 0.08

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Norepinephrine transporter inhibitor
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.05

    Interaction Types & Directionality:
    antagonist (inhibitory)

    Interaction Info:
    Direct Interaction yes
    Mechanism of Interaction Serotonin 2a (5-HT2a) receptor antagonist

    PMIDs:
    None found


  • Interaction Score: 0.02

    Interaction Types & Directionality:
    inhibitor (inhibitory)

    Interaction Info:
    Mechanism of Interaction Serotonin transporter inhibitor
    Direct Interaction yes

    PMIDs:
    None found